SCHEMBL18953702

SCHEMBL18953702

O=C(O)Nc1cccc(NS(=O)(=O)C2CC2)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTPS1 P17812 3/20 0.47
AAK1 Q2M2I8 7/20 0.47
GAK O14976 2/20 0.46
STK16 O75716 2/20 0.46
BMP2K Q9NSY1 2/20 0.46
HDAC4 P56524 1/20 0.46
OPRM1 P35372 1/20 0.45
GPR35 Q9HC97 1/20 0.43
USP2 O75604 1/20 0.43
LMNA P02545 1/20 0.43
GAA P10253 1/20 0.43
HPGD P15428 1/20 0.43
HTT P42858 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
HSD11B1 P28845 1/20 0.43
MAP2K7 O14733 1/20 0.43
MAP2K4 P45985 1/20 0.43
HSD17B1 P14061 2/20 0.42
HSD17B2 P37059 2/20 0.42
PTGS1 P23219 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18953568 0.83 HDAC4 (0.54) CTPS1HDAC4MAP2K4
SCHEMBL12407118 0.79 LMNA (0.52) AAK1OPRM1LMNAGAAHPGD
SCHEMBL28913080 0.78 LMNA (0.54) USP2LMNAGAAHPGDHTT
SCHEMBL3088255 0.78 HSD11B1 (0.57) AAK1HDAC4OPRM1SMN1; SMN2HSD11B1
SCHEMBL6850398 0.77 HDAC4 (0.56) HDAC4OPRM1MAP2K7MAP2K4PTGS1
SCHEMBL11858223 0.77 GPR35 (0.67) GPR35GAASMN1; SMN2
SCHEMBL23540320 0.77 CTPS1 (0.54) CTPS1OPRM1LMNAHTTSMN1; SMN2
SCHEMBL19329644 0.77 ALDH1A1 (0.65) GPR35HPGDHTTSMN1; SMN2HSD17B1
SCHEMBL3088257 0.77 HTR6 (0.56) AAK1GAKSTK16BMP2KHDAC4
SCHEMBL22619047 0.76 OPRM1 (0.48) AAK1GAKSTK16BMP2KHDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017098421-A1 BENZOTHIADIAZINE COMPOUNDS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2017-06-15 WO disclosed