SCHEMBL19003263

SCHEMBL19003263

CC(=O)Nc1cc(CN(C)S(=O)(=O)c2cccc(NC(=O)/C=C/c3ccc(Cl)s3)c2)cc(NC(=O)/C=C/c2ccc(Cl)s2)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 5/20 0.41
RAB9A P51151 3/20 0.41
NPC1 O15118 3/20 0.41
KEAP1 Q14145 1/20 0.41
NFE2L2 Q16236 1/20 0.41
MAPT P10636 8/20 0.41
MEN1 O00255 6/20 0.41
KMT2A Q03164 6/20 0.41
LMNA P02545 3/20 0.41
ALDH1A1 P00352 4/20 0.40
MAPK1 P28482 1/20 0.40
MITF O75030 1/20 0.40
HTT P42858 1/20 0.40
KCNJ6 P48051 2/20 0.39
KCNJ5 P48544 2/20 0.39
KCNJ3 P48549 2/20 0.39
POLB P06746 1/20 0.39
TP53 P04637 2/20 0.38
DHODH Q02127 1/20 0.38
NPSR1 Q6W5P4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19003240 0.83 MAPT (0.57) SMN1; SMN2RAB9ANPC1MAPTMEN1
SCHEMBL18985196 0.82 RAB9A (0.54) SMN1; SMN2RAB9ANPC1MAPTMEN1
SCHEMBL19003232 0.78 RAB9A (0.53) SMN1; SMN2RAB9ANPC1MAPTMEN1
SCHEMBL19003241 0.67 TGM2 (0.52) RAB9ANPC1MAPTMEN1KMT2A
SCHEMBL19003245 0.66 BCHE (0.58) SMN1; SMN2MAPTMEN1KMT2ALMNA
SCHEMBL19003252 0.66 RAB9A (0.53) SMN1; SMN2RAB9ANPC1MAPTMEN1
SCHEMBL12790129 0.66 KMT2A (0.64) SMN1; SMN2RAB9AMAPTMEN1KMT2A
SCHEMBL18985262 0.65 SMN1; SMN2 (0.51) SMN1; SMN2RAB9ANPC1MAPTMEN1
SCHEMBL18985260 0.65 SMN1; SMN2 (0.51) SMN1; SMN2RAB9ANPC1MAPTMEN1
SCHEMBL10788098 0.63 LMNA (0.68) SMN1; SMN2RAB9AMAPTLMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017102014-A1 PROPENAMIDE THIOPHENE DERIVATIVES AS FLAVIVIRUS INHIBITORS AND THEIR USE UNIVERSITE D'AIX-MARSEILLE (FR) 2017-06-22 WO disclosed