SCHEMBL19003345

SCHEMBL19003345

COc1cc(C)c(NC(=O)/C=C/c2ccc(Br)s2)cc1OC

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 6/20 0.47
KMT2A Q03164 6/20 0.47
MAPT P10636 5/20 0.47
SMN1; SMN2 Q16637 5/20 0.47
LMNA P02545 4/20 0.47
RAB9A P51151 4/20 0.47
MITF O75030 1/20 0.47
PAX8 Q06710 1/20 0.47
NPSR1 Q6W5P4 4/20 0.43
CYP3A4 P08684 3/20 0.43
NPC1 O15118 3/20 0.43
CYP1A2 P05177 2/20 0.43
CYP2C19 P33261 2/20 0.43
XBP1 P17861 1/20 0.43
TLR9 Q9NR96 1/20 0.43
HDAC3 O15379 2/20 0.42
HDAC4 P56524 2/20 0.42
HDAC1 Q13547 2/20 0.42
HDAC7 Q8WUI4 2/20 0.42
HDAC2 Q92769 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19003354 0.83 MMP1 (0.62) MEN1KMT2AMAPTSMN1; SMN2LMNA
SCHEMBL19003256 0.78 ALDH1A1 (0.64) MEN1KMT2AMAPTSMN1; SMN2LMNA
SCHEMBL19003347 0.77 CYP1A2 (0.54) MEN1KMT2AMAPTSMN1; SMN2LMNA
SCHEMBL9096395 0.76 MAPT (0.74) MEN1KMT2AMAPTSMN1; SMN2LMNA
SCHEMBL9096393 0.76 MAPT (0.74) MEN1KMT2AMAPTSMN1; SMN2LMNA
SCHEMBL19003274 0.75 MMP1 (0.58) MEN1KMT2AMAPTSMN1; SMN2LMNA
SCHEMBL19003351 0.72 LMNA (0.50) MEN1KMT2AMAPTSMN1; SMN2LMNA
SCHEMBL68058 0.72 CA12 (0.46) MEN1KMT2AMAPTSMN1; SMN2RAB9A
SCHEMBL68057 0.72 CA12 (0.46) MEN1KMT2AMAPTSMN1; SMN2RAB9A
SCHEMBL19003261 0.71 MMP1 (0.59) MEN1KMT2AMAPTSMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017102014-A1 PROPENAMIDE THIOPHENE DERIVATIVES AS FLAVIVIRUS INHIBITORS AND THEIR USE UNIVERSITE D'AIX-MARSEILLE (FR) 2017-06-22 WO disclosed