SCHEMBL1900979

SCHEMBL1900979

[c]1nn(C2CC2)cc1-c1ccccc1

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 7/20 0.35
DRD4 P21917 7/20 0.35
DRD3 P35462 6/20 0.35
SRC P12931 2/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33
CHRNB2 P17787 1/20 0.32
CHRNA4 P43681 1/20 0.32
BTK Q06187 1/20 0.32
HTR2A P28223 1/20 0.31
HTR2C P28335 1/20 0.31
HTR2B P41595 1/20 0.31
RIPK2 O43353 1/20 0.31
HRH3 Q9Y5N1 1/20 0.31
PDE10A Q9Y233 1/20 0.30
KCNH2 Q12809 2/20 0.30
SIGMAR1 Q99720 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL700238 0.69 PTGS2 (0.40)
SCHEMBL1851644 0.69 KMT2A (0.41)
SCHEMBL1900677 0.66 L3MBTL1 (0.36) DRD2
SCHEMBL1902680 0.66 KMT2A (0.34)
SCHEMBL1898425 0.66 CYP19A1 (0.32)
SCHEMBL6622485 0.55 CHRNB2 (0.43) CHRNB2CHRNA4HRH3
Biphenyl SCHEMBL547965 0.54 ALDH1A1 (0.90) SLC6A4
Biphenyl SCHEMBL21647236 0.54 ALDH1A1 (0.90) SLC6A4
Biphenyl SCHEMBL28376025 0.54 ALDH1A1 (0.60) SLC6A4
Biphenyl SCHEMBL1950563 0.54 ALDH1A1 (0.50) SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8455477-B2 Therapeutic compounds MERCK SHARP & DOHME CORP. (US) 2013-06-04 US disclosed
US-20110207711-A1 Therapeutic Compounds MSD K.K. (JP) 2011-08-25 US disclosed
EP-2320907-A1 THERAPEUTIC COMPOUNDS Merck & Co., Inc. (US) 2011-05-18 EP disclosed
WO-2010017047-A1 THERAPEUTIC COMPOUNDS MERCK & CO., INC. (US) 2010-02-11 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110207711-A1 Therapeutic Compounds WEE2, MARK3, WEE1 DRD2 2605/4885DRD4 3304/4885DRD3 2025/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.