SCHEMBL1902303

SCHEMBL1902303

CCC(C(=O)O)N1C(=O)Cc2cc(-c3ccc(F)c(F)c3)ccc21

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
BMPR1A P36894 13/20 0.39
ACVRL1 P37023 13/20 0.39
ACVR1 Q04771 13/20 0.39
BMPR1B O00238 12/20 0.39
TGFBR1 P36897 9/20 0.39
GRIN1 Q05586 2/20 0.36
GRIN2B Q13224 2/20 0.36
AKR1C3 P42330 1/20 0.35
AKR1C2 P52895 1/20 0.35
PDE5A O76074 1/20 0.35
NPY2R P49146 1/20 0.34
HRH3 Q9Y5N1 1/20 0.34
CYP11B1 P15538 1/20 0.34
CYP11B2 P19099 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16435034 0.89 CYP11B1 (0.40) GRIN1GRIN2BAKR1C3AKR1C2PDE5A
SCHEMBL1898876 0.89 BMPR1A (0.40) BMPR1AACVRL1ACVR1BMPR1BTGFBR1
SCHEMBL2003570 0.81 P2RX3 (0.42) PDE5A
SCHEMBL1896090 0.79 RXRA (0.40) BMPR1AACVRL1ACVR1BMPR1BTGFBR1
SCHEMBL16435091 0.74 HRH3 (0.41) AKR1C3AKR1C2HRH3
SCHEMBL12472190 0.72 LMNA (0.40)
SCHEMBL662686 0.72 LMNA (0.40)
SCHEMBL9108805 0.69 P2RX3 (0.43)
SCHEMBL3369814 0.69 DPP8 (0.40) BMPR1AACVRL1ACVR1BMPR1BTGFBR1
SCHEMBL9108017 0.68 PDE5A (0.49) PDE5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011056985-A2 SUBSTITUTED HETEROCYCLIC COMPOUNDS GILEAD SCIENCES, INC. (US) 2011-05-12 WO disclosed