SCHEMBL1896090

SCHEMBL1896090

CCC(C(=O)O)N1C(=O)Cc2cc(-c3cccc(OCF)c3)ccc21

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
RXRA P19793 1/20 0.40
RXRB P28702 1/20 0.40
BMPR1A P36894 6/20 0.37
ACVRL1 P37023 6/20 0.37
ACVR1 Q04771 6/20 0.37
BMPR1B O00238 5/20 0.37
TGFBR1 P36897 3/20 0.37
SLC13A5 Q86YT5 2/20 0.37
PTGS2 P35354 1/20 0.36
FFAR1 O14842 3/20 0.35
FFAR4 Q5NUL3 3/20 0.35
DHODH Q02127 3/20 0.35
NR4A2 P43354 2/20 0.35
HDAC1 Q13547 1/20 0.34
HDAC2 Q92769 1/20 0.34
PTPN1 P18031 1/20 0.34
AKR1C3 P42330 1/20 0.34
AKR1C2 P52895 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1898876 0.80 BMPR1A (0.40) BMPR1AACVRL1ACVR1BMPR1BTGFBR1
SCHEMBL1902303 0.79 BMPR1A (0.39) BMPR1AACVRL1ACVR1BMPR1BTGFBR1
SCHEMBL2003570 0.73 P2RX3 (0.42) HDAC1
SCHEMBL28853764 0.66 RXRA (0.73) RXRARXRBNR4A2HDAC1HDAC2
SCHEMBL9103481 0.65 NOTUM (0.40) PTGS2AKR1C3AKR1C2
SCHEMBL16435091 0.65 HRH3 (0.41) AKR1C3AKR1C2
SCHEMBL7467666 0.64 LTA4H (0.51) RXRARXRBFFAR1FFAR4NR4A2
SCHEMBL12472190 0.64 LMNA (0.40) HDAC1
SCHEMBL662686 0.64 LMNA (0.40) HDAC1
SCHEMBL3369814 0.64 DPP8 (0.40) BMPR1AACVRL1ACVR1BMPR1BTGFBR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011056985-A2 SUBSTITUTED HETEROCYCLIC COMPOUNDS GILEAD SCIENCES, INC. (US) 2011-05-12 WO disclosed