SCHEMBL19029520

SCHEMBL19029520

O=S(=O)(OCC1CC(F)(F)C1)c1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FFAR2 O15552 2/20 0.45
MAPK1 P28482 2/20 0.39
PARL Q9H300 1/20 0.38
GPR88 Q9GZN0 1/20 0.37
GBA1 P04062 1/20 0.37
TDP1 Q9NUW8 1/20 0.34
PRMT5 O14744 1/20 0.34
WDR77 Q9BQA1 1/20 0.34
ENPP3 O14638 1/20 0.34
CA2 P00918 1/20 0.34
ENPP1 P22413 1/20 0.34
ENPP2 Q13822 1/20 0.34
CA9 Q16790 1/20 0.34
ALDH1A1 P00352 2/20 0.33
HTR2A P28223 2/20 0.33
HTR2C P28335 2/20 0.33
HTR2B P41595 2/20 0.33
GAA P10253 1/20 0.33
MCOLN3 Q8TDD5 1/20 0.33
KDM4E B2RXH2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1864018 0.84 PLCG1 (0.38) FFAR2MAPK1CA2CA9ALDH1A1
SCHEMBL2304680 0.84 STAT3 (0.38) MAPK1CA2CA9ALDH1A1GAA
SCHEMBL6556991 0.77 GBA1 (0.43) FFAR2MAPK1PARLGBA1ENPP3
SCHEMBL28184784 0.76 ALDH1A1 (0.44) FFAR2MAPK1PARLGBA1ENPP3
SCHEMBL18372671 0.73 CYP2D6 (0.37) MAPK1ENPP3ENPP1ENPP2ALDH1A1
SCHEMBL23159147 0.71 FFAR2 (0.47) FFAR2MAPK1PARLGBA1PRMT5
SCHEMBL6555814 0.71 SMN1; SMN2 (0.41) MAPK1PARLGBA1ALDH1A1GAA
SCHEMBL13922018 0.71 ALDH1A1 (0.58) ALDH1A1GAAKDM4EHPGDKMT2A
SCHEMBL2796319 0.71 ARNT (0.39) ALDH1A1KDM4E
SCHEMBL9844160 0.70 PRMT5 (0.60) MAPK1PARLTDP1PRMT5WDR77

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107848953-B Fused ring gamma-amino acid derivative, preparation method and application thereof in medicine 四川海思科制药有限公司 2021-05-18 CN disclosed
CN-107848953-A Fused rings γ amino acid derivativges and preparation method thereof and application in medicine 四川海思科制药有限公司 2018-03-27 CN disclosed
WO-2017107907-A1 CONDENSED RING Γ-AMINO ACID DERIVATIVE AND PREPARATION METHOD AND MEDICAL USE THEREOF 四川海思科制药有限公司 2017-06-29 WO disclosed
WO-2017107907-A1 CONDENSED RING Γ-AMINO ACID DERIVATIVE AND PREPARATION METHOD AND MEDICAL USE THEREOF 四川海思科制药有限公司 2017-06-29 WO disclosed