SCHEMBL1907965

SCHEMBL1907965

O=C1Cc2cc(-c3cccc(C(F)(F)F)c3)ccc2N1

nearest known ligand 0.66

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 6/20 0.66
PGR P06401 2/20 0.63
CYP1A2 P05177 1/20 0.57
CYP11B1 P15538 1/20 0.57
CYP11B2 P19099 1/20 0.57
PDE3B Q13370 1/20 0.56
PDE3A Q14432 1/20 0.56
GRIA1 P42261 4/20 0.56
CACNG8 Q8WXS5 3/20 0.56
TDP2 O95551 1/20 0.55
PARP10 Q53GL7 1/20 0.53
PARP11 Q9NR21 1/20 0.53
GAA P10253 1/20 0.53
GRM2 Q14416 1/20 0.50
ASIC3 Q9UHC3 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1903306 0.88 KIF11 (0.80) KIF11PGRCYP1A2CYP11B1CYP11B2
SCHEMBL3315694 0.87 KIF11 (0.79) KIF11PGRCYP1A2CYP11B1CYP11B2
SCHEMBL25094235 0.86 PGR (0.63) KIF11PGRCYP1A2CYP11B1CYP11B2
SCHEMBL31492431 0.83 TDP2 (0.66) KIF11PDE3BPDE3ATDP2GAA
SCHEMBL578303 0.83 TDP2 (0.66) KIF11PDE3BPDE3ATDP2GAA
SCHEMBL3132725 0.81 PGR (0.73) KIF11PGRCYP1A2CYP11B1CYP11B2
SCHEMBL1900363 0.81 PGR (0.68) KIF11PGRCYP1A2CYP11B1CYP11B2
SCHEMBL1902698 0.80 KIF11 (0.59) KIF11PGRCYP1A2CYP11B1CYP11B2
SCHEMBL16208518 0.80 KIF11 (1.00) KIF11GAA
SCHEMBL3313408 0.79 KIF11 (0.62) KIF11TDP2PARP10PARP11ASIC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011056985-A2 SUBSTITUTED HETEROCYCLIC COMPOUNDS GILEAD SCIENCES, INC. (US) 2011-05-12 WO disclosed
US-4670566-A ANTIIFLAMMATORY AGENTS, ANTICOAGULANTS A. H. ROBINS COMPANY, INCORPORATED (US) 1987-06-02 US disclosed
US-4440785-A Methods of using 2-aminobiphenylacetic acids, esters, and metal salts thereof to treat inflammation A. H. ROBINS COMPANY, INC. (US) 1984-04-03 US disclosed