SCHEMBL19085984

SCHEMBL19085984

CC[C@@H](NC(=O)c1ccc2[nH]ncc2c1)C(=O)N1CCc2sc(C(=O)NCc3ccccc3)cc2C1

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 3/20 0.42
ROCK1 Q13464 2/20 0.42
KMT2A Q03164 2/20 0.41
KDM4E B2RXH2 1/20 0.41
MEN1 O00255 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
RXFP1 Q9HBX9 1/20 0.41
PRMT5 O14744 9/20 0.41
WDR77 Q9BQA1 9/20 0.41
HCRTR2 O43614 2/20 0.41
MAOB P27338 1/20 0.41
METTL3 Q86U44 1/20 0.40
AURKA O14965 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19085991 0.94 MAOB (0.42) ROCK2ROCK1KMT2AKDM4EMEN1
SCHEMBL19086985 0.94 PRMT5 (0.41) ROCK2ROCK1PRMT5WDR77MAOB
SCHEMBL19085995 0.93 METTL3 (0.41) ROCK2ROCK1KMT2AKDM4EMEN1
SCHEMBL19085983 0.93 ROCK2 (0.43) ROCK2ROCK1KMT2APRMT5WDR77
SCHEMBL19085994 0.92 ROCK2 (0.41) ROCK2ROCK1SMN1; SMN2PRMT5WDR77
SCHEMBL19085996 0.91 ROCK2 (0.53) ROCK2ROCK1PRMT5WDR77AURKA
SCHEMBL19086044 0.91 PRMT5 (0.40) ROCK2PRMT5WDR77MAOBMETTL3
SCHEMBL19085976 0.91 DDR2 (0.46) ROCK2ROCK1PRMT5WDR77MAOB
SCHEMBL19085985 0.90 PRMT5 (0.40) ROCK2ROCK1PRMT5WDR77METTL3
SCHEMBL19085999 0.90 TRPV1 (0.41) ROCK2ROCK1KMT2APRMT5WDR77

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017114275-A1 COMPOUND FOR INHIBITING ROCK, PREPARATION METHOD AND USE OF SAME 成都先导药物开发有限公司 2017-07-06 WO disclosed