SCHEMBL19145458

SCHEMBL19145458

C=C(NCC1CCN(C)CC1)c1ccc(N)cc1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 4/20 0.43
HDAC4 P56524 1/20 0.40
HDAC1 Q13547 1/20 0.39
HDAC2 Q92769 1/20 0.39
MAPT P10636 1/20 0.39
KDM1A O60341 1/20 0.38
MAOB P27338 1/20 0.38
MAP4K4 O95819 2/20 0.38
HDAC3 O15379 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
HTR4 Q13639 1/20 0.38
GSK3B P49841 1/20 0.38
EGLN1 Q9GZT9 1/20 0.38
NSD2 O96028 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23630645 0.83 NAMPT (0.60) NAMPTHDAC4HDAC1HDAC2MAP4K4
SCHEMBL19908021 0.81 HDAC3 (0.46) NAMPTHDAC4HDAC1HDAC2MAPT
SCHEMBL19145574 0.79 DRD1 (0.40) NAMPTHDAC4MAPTKDM1AMAOB
SCHEMBL12352674 0.79 ALDH1A1 (0.40) HDAC4HDAC1HDAC2MAPTHDAC3
SCHEMBL22326357 0.72 SIGMAR1 (0.50)
SCHEMBL12093537 0.70 MMP13 (0.61) NAMPTHDAC4HDAC1HDAC2HDAC3
SCHEMBL12090016 0.69 NAMPT (0.58) NAMPTHDAC4HDAC1HDAC2HDAC3
SCHEMBL2660481 0.69 NCF1 (0.42) NAMPTHDAC4HDAC1HDAC2MAPT
SCHEMBL16616770 0.69 NAMPT (0.67) NAMPTHDAC4EGLN1
SCHEMBL4040585 0.68 LMNA (0.53) MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017121444-A1 QUINOLIN-2-ONE DERIVATIVES MERCK PATENT GMBH (DE) 2017-07-20 WO disclosed