SCHEMBL1920182

SCHEMBL1920182

COc1ccc(S(=O)(=O)N(c2ccccc2C(F)(F)F)C(C(=O)O)c2cc(OC)ccc2S(=O)(=O)N(CC(=O)N2CCCC2c2ccc(F)cc2)c2ccccc2C(F)(F)F)cc1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CRHBP P24387 1/20 0.39
CRHR2 Q13324 1/20 0.39
KEAP1 Q14145 9/20 0.37
NFE2L2 Q16236 7/20 0.37
ALDH1A1 P00352 2/20 0.37
LMNA P02545 2/20 0.37
HSD17B10 Q99714 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
TSHR P16473 1/20 0.36
MAPT P10636 2/20 0.35
MAPK1 P28482 1/20 0.35
HTT P42858 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
SCD5 Q86SK9 1/20 0.35
KDM4E B2RXH2 1/20 0.34
OXTR P30559 1/20 0.34
AVPR1A P37288 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1921725 0.90 CRHBP (0.43) CRHBPCRHR2KEAP1NFE2L2ALDH1A1
SCHEMBL1921210 0.88 KEAP1 (0.41) CRHBPCRHR2KEAP1NFE2L2ALDH1A1
SCHEMBL1919868 0.87 CRHBP (0.48) CRHBPCRHR2KEAP1NFE2L2ALDH1A1
SCHEMBL1629345 0.87 CRHBP (0.49) CRHBPCRHR2KEAP1NFE2L2ALDH1A1
SCHEMBL1920350 0.86 MAPT (0.43) KEAP1NFE2L2ALDH1A1LMNAMAPT
SCHEMBL1920366 0.86 MDM4 (0.42) KEAP1NFE2L2ALDH1A1LMNAMAPT
SCHEMBL1919930 0.86 MDM4 (0.39) KEAP1NFE2L2ALDH1A1LMNAMAPT
SCHEMBL1920797 0.85 ALDH1A1 (0.42) KEAP1NFE2L2ALDH1A1LMNATSHR
SCHEMBL1920825 0.85 KMT2A (0.45) KEAP1NFE2L2ALDH1A1LMNAMAPT
SCHEMBL1920485 0.85 CRHBP (0.44) CRHBPCRHR2KEAP1NFE2L2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2245006-B1 SULFONAMIDES AS OREXIN ANTAGONISTS HOFFMANN LA ROCHE (CH) 2011-06-01 EP disclosed