SCHEMBL1920797

SCHEMBL1920797

COc1ccc(S(=O)(=O)N(c2cccc(C(F)(F)F)c2)C(C(=O)O)c2cc(OC)ccc2S(=O)(=O)N(CC(=O)N2CCCC2c2ccc(F)cc2)c2cccc(C(F)(F)F)c2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.42
USP2 O75604 1/20 0.42
HTT P42858 3/20 0.41
HPGD P15428 1/20 0.41
KMT2A Q03164 1/20 0.39
MAPT P10636 3/20 0.38
LMNA P02545 2/20 0.38
MAPK1 P28482 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
HCRTR1 O43613 1/20 0.37
HCRTR2 O43614 1/20 0.37
UTS2R Q9UKP6 1/20 0.37
KEAP1 Q14145 1/20 0.37
NFE2L2 Q16236 1/20 0.37
RORC P51449 4/20 0.37
HTR2A P28223 2/20 0.36
HTR2C P28335 2/20 0.36
HTR7 P34969 2/20 0.36
TSHR P16473 1/20 0.36
ALOX15 P16050 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1920177 0.96 HTT (0.44) ALDH1A1USP2HTTHPGDKMT2A
SCHEMBL1920825 0.94 KMT2A (0.45) ALDH1A1HTTKMT2AMAPTLMNA
SCHEMBL1920685 0.93 KMT2A (0.41) ALDH1A1HTTKMT2AMAPTLMNA
SCHEMBL1919930 0.92 MDM4 (0.39) ALDH1A1HTTKMT2AMAPTLMNA
SCHEMBL1920824 0.90 KMT2A (0.43) ALDH1A1HTTKMT2AMAPTLMNA
SCHEMBL1920366 0.90 MDM4 (0.42) ALDH1A1HTTKMT2AMAPTLMNA
SCHEMBL1920350 0.88 MAPT (0.43) ALDH1A1HTTKMT2AMAPTLMNA
SCHEMBL1630103 0.88 ALDH1A1 (0.52) ALDH1A1USP2HTTHPGDKMT2A
SCHEMBL1920294 0.86 MDM4 (0.48) ALDH1A1HTTKMT2AMAPTLMNA
SCHEMBL1920182 0.85 CRHBP (0.39) ALDH1A1HTTMAPTLMNAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2245006-B1 SULFONAMIDES AS OREXIN ANTAGONISTS HOFFMANN LA ROCHE (CH) 2011-06-01 EP disclosed