SCHEMBL1925175

SCHEMBL1925175

Nc1nc(NCc2ccncc2)nc(N(c2ccc(F)cc2)c2ccc(F)cc2)n1

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KCNH3 Q9ULD8 8/20 0.51
GPR68 Q15743 3/20 0.41
APP P05067 1/20 0.40
NPSR1 Q6W5P4 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA9 Q16790 1/20 0.38
HRH4 Q9H3N8 1/20 0.37
HRH3 Q9Y5N1 1/20 0.37
ADRA1D P25100 1/20 0.36
HTR2C P28335 1/20 0.36
HTR7 P34969 1/20 0.36
ADRA1A P35348 1/20 0.36
ADRA1B P35368 1/20 0.36
HTR6 P50406 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL536394 0.82 KCNH3 (0.52) KCNH3GPR68APPHTR2CHTR7
SCHEMBL29167130 0.77 CA1 (0.57) KCNH3GPR68APPNPSR1CA1
SCHEMBL29223873 0.75 CA1 (0.60) KCNH3GPR68APPNPSR1CA1
SCHEMBL1923563 0.69 KCNH3 (0.97) KCNH3
SCHEMBL1282106 0.68 ALDH1A1 (0.50) NPSR1
SCHEMBL5998625 0.67 KCNH3 (0.68) KCNH3NPSR1
SCHEMBL15721117 0.67 HTR7 (0.46) KCNH3CA1CA2CA9ADRA1D
SCHEMBL17173044 0.66 KCNH3 (0.51) KCNH3GPR68APPNPSR1CA1
SCHEMBL14869452 0.65 NPSR1 (0.59) GPR68APPNPSR1CA1CA2
SCHEMBL15720926 0.64 HTR7 (0.44) KCNH3CA1CA2CA9ADRA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1479397-B1 2,4,6-TRIAMINO-1,3,5-TRIAZINE DERIVATIVE ASTELLAS PHARMA INC (JP) 2011-06-08 EP claimed