SCHEMBL19257570

SCHEMBL19257570

COc1ccc(-c2ccc(-c3ccc(OC)c(C)c3)c(C#N)c2)c(CCC(=O)CO)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
XDH P47989 6/20 0.43
S1PR1 P21453 1/20 0.41
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
HSD17B10 Q99714 2/20 0.40
TP53 P04637 1/20 0.40
TBK1 Q9UHD2 1/20 0.38
MAPK8 P45983 2/20 0.37
MAPK9 P45984 2/20 0.37
PRKAB2 O43741 1/20 0.37
PRKAG1 P54619 1/20 0.37
PRKAA2 P54646 1/20 0.37
PRKAA1 Q13131 1/20 0.37
PRKAG3 Q9UGI9 1/20 0.37
PRKAG2 Q9UGJ0 1/20 0.37
PRKAB1 Q9Y478 1/20 0.37
MTNR1A P48039 1/20 0.36
MTNR1B P49286 1/20 0.36
MAPK10 P53779 1/20 0.36
KLKB1 P03952 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19209443 0.90 S1PR1 (0.51) XDHS1PR1HSD17B10
SCHEMBL19257720 0.87 XDH (0.42) XDHS1PR1NPC1RAB9AHSD17B10
SCHEMBL19209491 0.79 S1PR1 (0.46) XDHS1PR1NPC1RAB9AHSD17B10
SCHEMBL19209475 0.78 XDH (0.41) XDHS1PR1NPC1RAB9AHSD17B10
SCHEMBL15602073 0.78 RAB9A (0.44) NPC1RAB9AHSD17B10TP53MTNR1A
SCHEMBL1891972 0.78 POLB (0.50) S1PR1HSD17B10MTNR1AMTNR1B
SCHEMBL38659657 0.78 POLB (0.50) S1PR1HSD17B10MTNR1AMTNR1B
SCHEMBL19257588 0.78 HSD17B10 (0.43) NPC1RAB9AHSD17B10MTNR1AMTNR1B
SCHEMBL19209414 0.76 FFAR1 (0.50) XDHS1PR1MTNR1AMTNR1B
SCHEMBL38659061 0.75 MTNR1A (0.42) HSD17B10MTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017134146-A1 GPBP INHIBITORS AND USES AND SCALEABLE SYNTHESIS THEREOF FIBROSTATIN, S.L. (ES) 2017-08-10 WO disclosed