Leteprinim

Leteprinim

SCHEMBL194355

O=C(CCn1cnc2c(=O)[nH]cnc21)Nc1ccc(C(=O)O)cc1.[KH]

nearest known ligand 0.49

Full drug profile on Sugi Atlas →

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HPRT1 P00492 16/20 0.49
PNP P00491 2/20 0.46
LMNA P02545 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Leteprinim SCHEMBL358491 0.99 HPRT1 (0.50) HPRT1PNPLMNA
Leteprinim SCHEMBL6931317 0.98 HPRT1 (0.49) HPRT1PNP
Leteprinim SCHEMBL6935182 0.98 HPRT1 (0.49) HPRT1PNPLMNA
Leteprinim SCHEMBL194354 0.88 HPRT1 (0.48) HPRT1PNPLMNA
SCHEMBL1247298 0.85 GAA (0.54) HPRT1
SCHEMBL5258348 0.83 TK1 (0.54) HPRT1PNP
Leteprinim SCHEMBL358492 0.82 HSD17B10 (0.42) LMNA
SCHEMBL7684224 0.81 HPRT1 (0.49) HPRT1PNP
Hydrochloric Acid SCHEMBL7438455 0.80 HDAC3 (0.52) HPRT1LMNA
SCHEMBL7397072 0.78 HPRT1 (0.59) HPRT1PNP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 136 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1684784-A2 COMPOSITIONS OF A CYCLOOXYGENASE-2 SELECTIVE INHIBITOR AND A NEUROTROPHIC FACTOR-MODULATING AGENT FOR THE TREATMENT OF CENTRAL NERVOUS SYSTEM MEDIATED DISORDERS Pharmacia & Upjohn Company LLC (US) 2006-08-02 EP claimed
EP-1628532-A2 METHODS FOR THE PROTECTION OF MEMORY AND COGNITION Microbia, Inc. (US) 2006-03-01 EP claimed
US-20050148589-A1 Compositions of a cyclooxygenase-2 selective inhibitor and a neurotrophic factor-modulating agent for the treatment of central nervous system mediated disorders PHARMACIA & UPJOHN COMPANY LLC (US) 2005-07-07 US claimed
WO-2005046615-A2 COMPOSITIONS FOR TREATMENT OF CENTRAL NERVOUS SYSTEM MEDIATED DISORDERS PHARMACIA & UPJOHN COMPANY LLC (US) 2005-05-26 WO claimed
US-20050020945-A1 Acoustically-aided cerebrospinal-fluid manipulation for neurodegenerative disease therapy TOSAYA CAROL A (US) 2005-01-27 US claimed
US-20050004104-A1 Methods for the protection of memory and cognition IRONWOOD PHARMACEUTICALS, INC. 2005-01-06 US claimed
WO-2004108085-A2 METHODS FOR THE PROTECTION OF MEMORY AND COGNITION MICROBIA, INC. (US) 2004-12-16 WO claimed
US-20040049134-A1 System and methods for treatment of alzheimer's and other deposition-related disorders of the brain TOSAYA CAROL A (US) 2004-03-11 US claimed
EP-3157408-B1 DEVICES TO PROVIDE HANDS FREE SCLERAL DEPRESSION DURING OPHTHALMIC PROCEDURES ALCON INC (CH) 2026-03-25 EP disclosed
EP-4714407-A2 DEVICES TO PROVIDE HANDS FREE SCLERAL DEPRESSION DURING OPHTHALMIC PROCEDURES Alcon Inc. (CH) 2026-03-25 EP disclosed
US-20250057694-A1 DEVICES AND METHODS TO PROVIDE HANDS FREE SCLERAL DEPRESSION AND ILLUMINATION DURING OPHTHALMIC PROCEDURES Ganihand, LLC (US) 2025-02-20 US disclosed
US-11266395-B2 Devices and methods to provide hands free scleral depression during ophthalmic procedures Ganihand, LLC (US) 2022-03-08 US disclosed
CN-110290781-A The dosage form of stomach and intestine privileged site control release 南京三迭纪医药科技有限公司 2019-09-27 CN disclosed
CN-107847398-B Control the pharmaceutical dosage form of release 南京三迭纪医药科技有限公司 2019-05-07 CN disclosed
US-20020040031-A1 Methods for prevention of accumulation of amyloid beta peptide in the central nervous system NEO THERAPEUTICS, INC. 2002-04-04 US disclosed
WO-2002004449-A2 METHODS FOR TREATMENT OF CONDITIONS AFFECTED BY ACTIVITY OF MULTIDRUG TRANSPORTERS NEOTHERAPEUTICS, INC. (US) 2002-01-17 WO disclosed
WO-2002004450-A2 METHODS FOR PREVENTION OF ACCUMULATION OF AMYLOID BETA PEPTIDE IN THE CENTRAL NERVOUS SYSTEM NEOTHERAPEUTICS, INC. (US) 2002-01-17 WO disclosed
WO-2002004451-A2 METHODS FOR STIMULATION OF SYNTHESIS OF SYNAPTOPHYSIN IN THE CENTRAL NERVOUS SYSTEM NEOTHERAPEUTICS, INC. (US) 2002-01-17 WO disclosed
WO-2002004452-A2 METHODS FOR TREATMENT OF DISEASE-INDUCED PERIPHERAL NEUROPATHY AND RELATED CONDITIONS NEOTHERAPEUTICS, INC. (US) 2002-01-17 WO disclosed
WO-2002004448-A2 METHODS FOR TREATMENT OF DRUG-INDUCED PERIPHERAL NEUROPATHY AND RELATED CONDITIONS NEOTHERAPEUTICS, INC. (US) 2002-01-17 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050004104-A1 Methods for the protection of memory and cognition PTGES2, PTGS2, PTGS1 HPRT1 983/4885PNP 3281/4885LMNA 3639/4885
US-20050148589-A1 Compositions of a cyclooxygenase-2 selective inhibitor and a neurotrophic factor-modulating agent for the treatment of central nervous system mediated disorders BDNF, NTRK2, NGF HPRT1 3707/4885PNP 2597/4885LMNA 3783/4885
US-20020040031-A1 Methods for prevention of accumulation of amyloid beta peptide in the central nervous system APP, BACE1, SARNP HPRT1 10/4885PNP 9/4885LMNA 623/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.