Leteprinim

Leteprinim

SCHEMBL358491

O=C(CCn1cnc2c(=O)[nH]cnc21)Nc1ccc(C(=O)O)cc1

nearest known ligand 0.50

Full drug profile on Sugi Atlas →

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HPRT1 P00492 16/20 0.50
PNP P00491 2/20 0.47
LMNA P02545 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Leteprinim SCHEMBL194355 0.99 HPRT1 (0.49) HPRT1PNPLMNA
Leteprinim SCHEMBL6931317 0.99 HPRT1 (0.49) HPRT1PNP
Leteprinim SCHEMBL6935182 0.99 HPRT1 (0.49) HPRT1PNPLMNA
Leteprinim SCHEMBL194354 0.89 HPRT1 (0.48) HPRT1PNPLMNA
SCHEMBL1247298 0.86 GAA (0.54) HPRT1
SCHEMBL5258348 0.84 TK1 (0.54) HPRT1PNP
Leteprinim SCHEMBL358492 0.83 HSD17B10 (0.42) LMNA
SCHEMBL7684224 0.82 HPRT1 (0.49) HPRT1PNP
Hydrochloric Acid SCHEMBL7438455 0.81 HDAC3 (0.52) HPRT1LMNA
SCHEMBL7397072 0.79 HPRT1 (0.59) HPRT1PNP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 790 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024258996-A1 OCULAR DRUG DELIVERY BAYLOR COLLEGE OF MEDICINE (US) 2024-12-19 WO claimed
CN-112469406-A Use of stearic acid for preventing or treating pulmonary fibrosis 财团法人峨山社会福祉财团 2021-03-09 CN claimed
US-20150328323-A1 Nitric Oxide Releasing Produgs of Therapeutic Agents SATYAM APPARAO (IN) 2015-11-19 US claimed
US-9016221-B2 Surface topographies for non-toxic bioadhesion control UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2015-04-28 US claimed
WO-2014111957-A1 NITRIC OXIDE RELEASING PRODRUGS OF THERAPEUTIC AGENTS SATYAM APPARAO (IN) 2014-07-24 WO claimed
US-20120276019-A1 TISSUE KALLIKREIN FOR THE TREATMENT OF PARKINSON'S DISEASE DIAMEDICA INC. (CA) 2012-11-01 US claimed
US-20110150781-A1 TISSUE KALLIKREIN FOR THE TREATMENT OF PARKINSON'S DISEASE DIAMEDICA INC. (CA) 2011-06-23 US claimed
EP-2320939-A1 TISSUE KALLIKREIN FOR THE TREATMENT OF PARKINSON'S DISEASE Sanomune Inc. (CA) 2011-05-18 EP claimed
EP-1790344-B1 Methods for treatment of disease-induced peripheral neuropathy and related conditions SPECTRUM PHARMACEUTICALS INC (US) 2011-02-23 EP claimed
US-20100226943-A1 SURFACE TOPOGRAPHIES FOR NON-TOXIC BIOADHESION CONTROL UNIVERSITY OF FLORIDA (US) 2010-09-09 US claimed
WO-2001036419-A1 USE OF 9-SUBSTITUTED HYPOXANTHINE DERIVATIVES TO STIMULATE REGENERATION OF NERVOUS TISSUE NEOTHERAPEUTICS, INC. (US) 2001-05-25 WO claimed
WO-2001028545-A2 USE OF CARBON MONOXIDE DEPENDENT GUANYLYL CYCLASE MODIFIERS TO STIMULATE NEURITOGENESIS NEOTHERAPEUTICS, INC. (US) 2001-04-26 WO claimed
US-6027936-A ADMINISTERING AMOUNT OF AT LEAST ONE MODULATING PURINE DERIVATIVE TO A MAMMAL FOR SELECTIVE INDUCTION OF GENE EXPRESSION OF MOLECULE THAT STIMULATES NEURITOGENESIS; TREATMENT AND PROPHYLAXIS FOR NERVOUS SYSTEM DISORDERS SPECTRUM PHARMACEUTICALS, INC. 2000-02-22 US claimed
EP-0772440-A4 CARBON MONOXIDE DEPENDENT GUANYLYL CYCLASE MODIFIERS GLASKY ALVIN J (US) 1999-05-19 EP claimed
US-5801184-A Carbon monoxide dependent guanylyl cyclase modifiers and methods of use SPECTRUM PHARMACEUTICALS, INC. 1998-09-01 US claimed
EP-0522082-B1 MULTI-FUNCTIONAL PHARMACEUTICAL COMPOUNDS AND METHODS OF USE GLASKY ALVIN J (US) 1997-07-02 EP claimed
EP-0772440-A1 CARBON MONOXIDE DEPENDENT GUANYLYL CYCLASE MODIFIERS GLASKY, Alvin J. (US) 1997-05-14 EP claimed
WO-1996003125-A1 CARBON MONOXIDE DEPENDENT GUANYLYL CYCLASE MODIFIERS GLASKY ALVIN J (US) 1996-02-08 WO claimed
US-5447939-A Purine derivatives used for long term modification of neural activity in mammals, for treatment of mammalian neurological diseases, and for inducing long term changes in membrane potential of mammalian neuron SPECTRUM PHARMACEUTICALS, INC. 1995-09-05 US claimed
US-5091432-A Synergistic SPECTRUM PHARMACEUTICALS, INC. 1992-02-25 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150328323-A1 Nitric Oxide Releasing Produgs of Therapeutic Agents NOS2, NOS1, PTGIS HPRT1 848/4885PNP 166/4885LMNA 1146/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.