SCHEMBL19494263

SCHEMBL19494263

C=N/C(=C\CC)N1CCOCC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.38
TSHR P16473 2/20 0.38
L3MBTL1 Q9Y468 1/20 0.36
MGLL Q99685 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
ALDH1A1 P00352 2/20 0.35
PDK1 Q15118 2/20 0.35
PDK2 Q15119 2/20 0.35
PDK3 Q15120 2/20 0.35
FAAH O00519 1/20 0.35
PHGDH O43175 1/20 0.35
ALDH2 P05091 1/20 0.35
RECQL P46063 1/20 0.35
MAPT P10636 1/20 0.35
POLB P06746 3/20 0.34
LMNA P02545 3/20 0.33
CA12 O43570 2/20 0.32
CA1 P00915 2/20 0.32
CA9 Q16790 2/20 0.32
CA2 P00918 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24318148 0.80 SMN1; SMN2 (0.40) HTTTSHRL3MBTL1MGLLSMN1; SMN2
SCHEMBL24497941 0.74 MAPT (0.37) HTTTSHRL3MBTL1MGLLSMN1; SMN2
SCHEMBL8553865 0.72 SMN1; SMN2 (0.45) HTTTSHRL3MBTL1MGLLSMN1; SMN2
SCHEMBL8553868 0.72 SMN1; SMN2 (0.45) HTTTSHRL3MBTL1MGLLSMN1; SMN2
SCHEMBL20120036 0.72 MAPT (0.43) HTTTSHRL3MBTL1MGLLSMN1; SMN2
SCHEMBL19286446 0.71 LMNA (0.38) HTTL3MBTL1MGLLSMN1; SMN2ALDH1A1
SCHEMBL5274271 0.71 HTT (0.46) HTTTSHRL3MBTL1MGLLSMN1; SMN2
SCHEMBL19566668 0.70 SMN1; SMN2 (0.36) HTTL3MBTL1MGLLSMN1; SMN2ALDH1A1
SCHEMBL24313179 0.70 PDK1 (0.36) HTTPDK1PDK2PDK3LMNA
SCHEMBL21504068 0.69 L3MBTL1 (0.42) HTTTSHRL3MBTL1MGLLSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3235816-B1 2-MORPHOLIN-4,6-DISUBSTITUTED PYRIMIDINE DERIVATIVE, AND PREPARATION METHOD AND PHARMACEUTICAL USE THEREOF SHANGHAI HAIYAN PHARMACEUTICAL TECH CO LTD (CN) 2020-02-12 EP disclosed
EP-3235816-A1 2-MORPHOLIN-4,6-DISUBSTITUTED PYRIMIDINE DERIVATIVE, AND PREPARATION METHOD AND PHARMACEUTICAL USE THEREOF Shanghai Haiyan Pharmaceutical Technology Co., Ltd. (CN) 2017-10-25 EP disclosed