SCHEMBL19615959

SCHEMBL19615959

CC(O)(Cn1cncn1)c1cc(Oc2ccc(Cl)cc2)ccc1C(F)(F)F

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 10/20 0.47
ALDH1A1 P00352 2/20 0.47
KMT2A Q03164 1/20 0.46
CYP2C9 P11712 8/20 0.41
CYP2C19 P33261 8/20 0.41
CYP19A1 P11511 3/20 0.41
HSP90AA1 P07900 3/20 0.41
LMNA P02545 1/20 0.41
CYP11B1 P15538 1/20 0.41
CYP11B2 P19099 1/20 0.41
ADRA1A P35348 1/20 0.41
CYP51A1 Q16850 1/20 0.41
AR P10275 2/20 0.41
CYP1A2 P05177 3/20 0.38
CYP2D6 P10635 3/20 0.38
KCNH2 Q12809 2/20 0.38
TSHR P16473 1/20 0.38
POLB P06746 1/20 0.37
KDM4E B2RXH2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29427653 1.00 CYP3A4 (0.47) CYP3A4ALDH1A1KMT2ACYP2C9CYP2C19
SCHEMBL14645411 0.96 CYP3A4 (0.47) CYP3A4ALDH1A1KMT2ACYP2C9CYP2C19
SCHEMBL29359684 0.96 CYP3A4 (0.47) CYP3A4ALDH1A1KMT2ACYP2C9CYP2C19
SCHEMBL29133281 0.96 CYP3A4 (0.47) CYP3A4ALDH1A1KMT2ACYP2C9CYP2C19
SCHEMBL29363144 0.96 CYP3A4 (0.47) CYP3A4ALDH1A1KMT2ACYP2C9CYP2C19
SCHEMBL15821868 0.96 CYP3A4 (0.47) CYP3A4ALDH1A1KMT2ACYP2C9CYP2C19
SCHEMBL15832616 0.96 CYP3A4 (0.47) CYP3A4ALDH1A1KMT2ACYP2C9CYP2C19
SCHEMBL29362708 0.96 CYP3A4 (0.47) CYP3A4ALDH1A1KMT2ACYP2C9CYP2C19
SCHEMBL29133282 0.96 CYP3A4 (0.47) CYP3A4ALDH1A1KMT2ACYP2C9CYP2C19
SCHEMBL14637517 0.88 CYP3A4 (0.49) CYP3A4ALDH1A1KMT2ACYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 35 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230126361-A1 METHODS OF CONTROLLING OR PREVENTING INFESTATION OF PLANTS BY THE PHYTOPATHOGENIC MICROORGANISM CORYNESPORA CASSIICOLA, CERCOSPORA SOJINA AND/OR CERCOSPORA KIKUCHII SYNGENTA CROP PROTECTION AG (CH) 2023-04-27 US claimed
US-11154058-B2 Fungicidal compositions SYNGENTA PARTICIPATIONS AG (CH) 2021-10-26 US claimed
US-20200329703-A1 FUNGICIDAL COMPOSITIONS SYNGENTA PARTICIPATIONS AG (CH) 2020-10-22 US claimed
EP-3717479-B1 MICROBIOCIDAL THIAZOLE DERIVATIVES SYNGENTA PARTICIPATIONS AG (CH) 2023-07-05 EP disclosed
US-20230126361-A1 METHODS OF CONTROLLING OR PREVENTING INFESTATION OF PLANTS BY THE PHYTOPATHOGENIC MICROORGANISM CORYNESPORA CASSIICOLA, CERCOSPORA SOJINA AND/OR CERCOSPORA KIKUCHII SYNGENTA CROP PROTECTION AG (CH) 2023-04-27 US disclosed
US-20230112306-A1 METHODS OF CONTROLLING OR PREVENTING INFESTATION OF SOYBEAN PLANTS BY THE PHYTOPATHOGENIC MICROORGANISM CORYNESPORA CASSIICOLA SYNGENTA CROP PROTECTION AG (CH) 2023-04-13 US disclosed
US-20230111656-A1 METHODS OF CONTROLLING OR PREVENTING INFESTATION OF SOYBEAN PLANTS BY THE PHYTOPATHOGENIC MICROORGANISM CORYNESPORA CASSIICOLA SYNGENTA CROP PROTECTION AG (CH) 2023-04-13 US disclosed
EP-3692029-B1 MICROBIOCIDAL PICOLINAMIDE DERIVATIVES SYNGENTA PARTICIPATIONS AG (CH) 2023-04-12 EP disclosed
EP-3710429-B1 MICROBIOCIDAL PICOLINAMIDE DERIVATIVES SYNGENTA PARTICIPATIONS AG (CH) 2023-04-05 EP disclosed
EP-3853207-B1 MICROBIOCIDAL QUINOLINE CARBOXAMIDE DERIVATIVES SYNGENTA CROP PROTECTION AG (CH) 2022-10-19 EP disclosed
EP-3683213-B1 INTERMEDIATE FOR THE PREPARATION OF MICROBIOCIDAL HETEROBICYCLIC DERIVATIVES SYNGENTA PARTICIPATIONS AG (CH) 2022-10-12 EP disclosed
EP-3582616-B1 FUNGICIDAL COMPOSITIONS SYNGENTA PARTICIPATIONS AG (CH) 2020-12-16 EP disclosed
US-20200329703-A1 FUNGICIDAL COMPOSITIONS SYNGENTA PARTICIPATIONS AG (CH) 2020-10-22 US disclosed
US-20200207692-A1 PROCESS FOR THE PREPARATION OF SUBSTITUTED PHENOXYPHENYL ALCOHOLS BASF SE (DE) 2020-07-02 US disclosed
EP-3274343-B1 MICROBIOCIDAL HETEROBICYCLIC DERIVATIVES SYNGENTA PARTICIPATIONS AG (CH) 2020-03-04 EP disclosed
EP-3606913-A1 MICROBIOCIDAL OXADIAZOLE DERIVATIVES Syngenta Participations AG (CH) 2020-02-12 EP disclosed
EP-3458446-A1 MICROBIOCIDAL OXADIAZOLE DERIVATIVES Syngenta Participations AG (CH) 2019-03-27 EP disclosed
WO-2018184982-A1 MICROBIOCIDAL OXADIAZOLE DERIVATIVES SYNGENTA PARTICIPATIONS AG (CH) 2018-10-11 WO disclosed
WO-2018185013-A1 MICROBIOCIDAL OXADIAZOLE DERIVATIVES SYNGENTA PARTICIPATIONS AG (CH) 2018-10-11 WO disclosed
WO-2017198852-A1 MICROBIOCIDAL OXADIAZOLE DERIVATIVES SYNGENTA PARTICIPATIONS AG (CH) 2017-11-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200329703-A1 FUNGICIDAL COMPOSITIONS PFAS, NAT1, PAH CYP3A4 53/4885ALDH1A1 901/4885KMT2A 1375/4885
US-11154058-B2 Fungicidal compositions PFAS, NAT1, PAH CYP3A4 53/4885ALDH1A1 901/4885KMT2A 1375/4885
US-20200207692-A1 PROCESS FOR THE PREPARATION OF SUBSTITUTED PHENOXYPHENYL ALCOHOLS ADH1C, ADH1A, ADH5 CYP3A4 98/4885ALDH1A1 169/4885KMT2A 2070/4885
US-20230112306-A1 METHODS OF CONTROLLING OR PREVENTING INFESTATION OF SOYBEAN PLANTS BY THE PHYTOPATHOGENIC MICROORGANISM CORYNESPORA CASSIICOLA NIT2, NSFL1C, NOS2 CYP3A4 754/4885ALDH1A1 3123/4885KMT2A 3148/4885
US-20230126361-A1 METHODS OF CONTROLLING OR PREVENTING INFESTATION OF PLANTS BY THE PHYTOPATHOGENIC MICROORGANISM CORYNESPORA CASSIICOLA, CERCOSPORA SOJINA AND/OR CERCOSPORA KIKUCHII DPM1, SACM1L, SYNJ1 CYP3A4 731/4885ALDH1A1 780/4885KMT2A 896/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.