SCHEMBL19626577

SCHEMBL19626577

CC(C)(C)c1nc(-c2cccc(C(F)(F)F)c2)cs1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.53
MEN1 O00255 2/20 0.53
KMT2A Q03164 2/20 0.53
KDM4E B2RXH2 2/20 0.53
AR P10275 1/20 0.53
ADAM17 P78536 1/20 0.50
CFTR P13569 2/20 0.49
CASP3 P42574 1/20 0.48
CASP7 P55210 1/20 0.48
CASP8 Q14790 1/20 0.48
KDM1A O60341 1/20 0.47
CTSS P25774 1/20 0.47
LTA4H P09960 1/20 0.46
IDO1 P14902 1/20 0.46
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
GABRA1 P14867 1/20 0.45
HPGD P15428 1/20 0.45
GABRG2 P18507 1/20 0.45
GABRB3 P28472 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2405752 0.85 RECQL (0.60) ALDH1A1MEN1KMT2AKDM4EAR
SCHEMBL19625325 0.82 KDM4E (0.62) ALDH1A1MEN1KMT2AKDM4ECYP1A2
SCHEMBL13118019 0.81 LTA4H (0.54) ALDH1A1MEN1KMT2AKDM4EKDM1A
SCHEMBL12868318 0.81 ATP4A (0.55) ALDH1A1MEN1KMT2ACASP3LTA4H
SCHEMBL1198896 0.80 ALDH1A1 (0.56) ALDH1A1MEN1KMT2AKDM4EAR
SCHEMBL28743338 0.80 ALDH1A1 (0.71) ALDH1A1MEN1KMT2AKDM4EAR
SCHEMBL474410 0.80 LTA4H (0.67) ALDH1A1MEN1KMT2AKDM4EAR
SCHEMBL19625426 0.79 TRPA1 (0.42) MEN1KMT2AKDM4EARADAM17
SCHEMBL19625389 0.79 SCN9A (0.51) CTSSKITTRPA1
Bromide SCHEMBL8357468 0.79 LTA4H (0.65) ALDH1A1MEN1KMT2AKDM4EAR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10472360-B2 Purine diones as Wnt pathway modulators AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2019-11-12 US disclosed
US-20170334912-A1 Purine Diones As Wnt Pathway Modulators AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2017-11-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170334912-A1 Purine Diones As Wnt Pathway Modulators WNT1, WNT3A, CTNNB1 ALDH1A1 1166/4885MEN1 4625/4885KMT2A 3504/4885
US-10472360-B2 Purine diones as Wnt pathway modulators WNT1, WNT3A, CTNNB1 ALDH1A1 1166/4885MEN1 4625/4885KMT2A 3504/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.