SCHEMBL1964639

SCHEMBL1964639

Cc1cc(C=O)ccc1-c1nnc(-c2ccccc2C(N)=O)s1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.39
NPC1 O15118 3/20 0.39
RAB9A P51151 2/20 0.39
LMNA P02545 2/20 0.39
CSNK1A1 P48729 1/20 0.39
TYRO3 Q06418 1/20 0.39
DYRK1B Q9Y463 1/20 0.39
BCAT2 O15382 1/20 0.37
PTGER3 P43115 1/20 0.36
TRPV1 Q8NER1 1/20 0.35
KDM4E B2RXH2 1/20 0.35
USP2 O75604 1/20 0.35
GAA P10253 1/20 0.35
HPGD P15428 1/20 0.35
MYC P01106 1/20 0.35
CTSA P10619 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34
DDX3X O00571 1/20 0.34
EIF4E P06730 1/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1968589 0.89 ALDH1A1 (0.40) ALDH1A1NPC1RAB9ALMNACSNK1A1
SCHEMBL1965022 0.82 BCAT2 (0.44) NPC1RAB9ACSNK1A1TYRO3DYRK1B
SCHEMBL1966405 0.81 BCAT2 (0.40) ALDH1A1NPC1RAB9ALMNACSNK1A1
SCHEMBL1964640 0.74 SMN1; SMN2 (0.55) ALDH1A1NPC1RAB9ALMNAPTGER3
SCHEMBL1968944 0.73 BCAT2 (0.43) NPC1RAB9ACSNK1A1TYRO3DYRK1B
SCHEMBL17158372 0.73 MYC (0.51) ALDH1A1NPC1RAB9ALMNAKDM4E
SCHEMBL18584726 0.73 BCAT2 (0.61) NPC1RAB9ACSNK1A1TYRO3DYRK1B
SCHEMBL1800318 0.70 PARP10 (0.44) ALDH1A1RAB9AKDM4EUSP2GAA
SCHEMBL15330096 0.68 CTNNB1 (0.49) ALDH1A1NPC1RAB9ALMNAKDM4E
SCHEMBL15650835 0.67 TDP1 (0.43) ALDH1A1RAB9AKDM4EUSP2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2334670-A1 NEW 2-AMIDOTHIADIAZOLE DERIVATIVES Almirall S.A. (ES) 2011-06-22 EP disclosed