SCHEMBL1968944

SCHEMBL1968944

C=Cc1ccc(-c2nnc(-c3ccccc3C(N)=O)s2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCAT2 O15382 1/20 0.43
PTGES O14684 1/20 0.40
ALOX5 P09917 1/20 0.40
CSNK1A1 P48729 1/20 0.39
TYRO3 Q06418 1/20 0.39
DYRK1B Q9Y463 1/20 0.39
PARP1 P09874 1/20 0.39
TRPV1 Q8NER1 1/20 0.37
NPC1 O15118 5/20 0.36
RAB9A P51151 5/20 0.36
DDX3X O00571 3/20 0.36
ROCK2 O75116 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
KDM4E B2RXH2 1/20 0.35
EIF4E P06730 1/20 0.35
CSNK2A2 P19784 1/20 0.35
CSNK2B P67870 1/20 0.35
CSNK2A1 P68400 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1965022 0.88 BCAT2 (0.44) BCAT2PTGESALOX5CSNK1A1TYRO3
SCHEMBL18584726 0.84 BCAT2 (0.61) BCAT2PTGESALOX5CSNK1A1TYRO3
SCHEMBL1968589 0.83 ALDH1A1 (0.40) BCAT2CSNK1A1TYRO3DYRK1BPARP1
SCHEMBL1966405 0.73 BCAT2 (0.40) BCAT2PTGESALOX5CSNK1A1TYRO3
SCHEMBL11611572 0.72 NPC1 (0.56) NPC1RAB9ADDX3XMEN1KMT2A
SCHEMBL27947437 0.71 BCAT2 (0.43) BCAT2CSNK1A1TYRO3DYRK1BPARP1
SCHEMBL1968945 0.68 CSNK2A2 (0.71) NPC1RAB9ADDX3XMEN1KMT2A
SCHEMBL25353879 0.67 HNF4A (0.49) BCAT2NPC1RAB9AMEN1KMT2A
SCHEMBL5878337 0.67 BCAT2 (0.87) BCAT2CSNK1A1TYRO3DYRK1BPARP1
SCHEMBL28054906 0.67 BCAT2 (0.56) BCAT2CSNK1A1TYRO3DYRK1BPARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2334670-A1 NEW 2-AMIDOTHIADIAZOLE DERIVATIVES Almirall S.A. (ES) 2011-06-22 EP disclosed