SCHEMBL19687558

SCHEMBL19687558

CCCOCCOCCOCCOc1cccnc1N(C)C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.40
MAPT P10636 4/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
MAPK1 P28482 1/20 0.40
CYP2C19 P33261 1/20 0.40
PDE5A O76074 3/20 0.40
PDE4A P27815 3/20 0.40
PDE4B Q07343 3/20 0.40
PDE4C Q08493 3/20 0.40
PDE4D Q08499 3/20 0.40
ADRB2 P07550 1/20 0.39
ADRB1 P08588 1/20 0.39
LMNA P02545 5/20 0.39
ALDH1A1 P00352 6/20 0.38
HTT P42858 2/20 0.38
GRM5 P41594 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
TDP1 Q9NUW8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19687559 0.86 KDM4E (0.40) KDM4EMAPTCYP1A2CYP3A4CYP2C9
SCHEMBL19631332 0.86 KDM4E (0.41) KDM4EMAPTCYP1A2CYP3A4CYP2C9
SCHEMBL25914790 0.81 CHRNB2 (0.43) KDM4EMAPTCYP1A2CYP3A4CYP2C9
SCHEMBL21100993 0.81 CHRNB2 (0.43) KDM4EMAPTCYP1A2CYP3A4CYP2C9
SCHEMBL17784960 0.80 LMNA (0.37) KDM4EMAPTCYP1A2CYP3A4CYP2C9
SCHEMBL28015202 0.80 GRM5 (0.46) KDM4EMAPTPDE5ALMNAALDH1A1
SCHEMBL19342481 0.79 CHRNB2 (0.47) KDM4EMAPTCYP1A2CYP3A4CYP2C9
SCHEMBL22736821 0.78 PRMT5 (0.35) KDM4EMAPTPDE5APDE4APDE4B
SCHEMBL21500781 0.75 ALDH1A1 (0.36) KDM4EMAPTMAPK1LMNAALDH1A1
SCHEMBL19687565 0.74 LMNA (0.40) KDM4EMAPTCYP1A2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017210335-A1 IMAGING METHODS USING 18F-RADIOLABELED BIOLOGICS BRISTOL-MYERS SQUIBB COMPANY (US) 2017-12-07 WO disclosed