SCHEMBL19781568

SCHEMBL19781568

CCc1cc2ncc(C)n2cc1Br

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 1/20 0.33
NOS1 P29475 1/20 0.33
NOS2 P35228 1/20 0.33
KDM4E B2RXH2 3/20 0.32
RAB9A P51151 2/20 0.32
POLB P06746 1/20 0.32
NR4A1 P22736 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
ESR2 Q92731 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
PRMT5 O14744 2/20 0.31
WDR77 Q9BQA1 2/20 0.31
SCN9A Q15858 1/20 0.31
ALDH1A1 P00352 2/20 0.31
GLA P06280 2/20 0.31
GAA P10253 2/20 0.31
HPGD P15428 2/20 0.31
NPC1 O15118 1/20 0.31
TP53 P04637 1/20 0.31
CYP1A2 P05177 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19781784 0.79 TRPA1 (0.34) KDM4ERAB9AALDH1A1NPC1TGFBR1
SCHEMBL1913167 0.77 TGFBR1 (0.44) KDM4ERAB9APOLBNPSR1ALDH1A1
SCHEMBL20985980 0.77 TGFBR1 (0.34) KDM4ERAB9AALDH1A1NPC1TGFBR1
SCHEMBL24460464 0.73 PIK3CA (0.39) KDM4ERAB9AALDH1A1HPGDNPC1
SCHEMBL20049572 0.72 NPC1 (0.33) RAB9APRMT5WDR77NPC1TGFBR1
SCHEMBL20049571 0.72 PRMT5 (0.32) PRMT5WDR77TGFBR1
SCHEMBL22072385 0.72 GABRA1 (0.37) KDM4ERAB9ANPSR1ALDH1A1NPC1
SCHEMBL24460481 0.71 POLB (0.39) KDM4ERAB9APOLBNPSR1TDP1
SCHEMBL1913154 0.68 KEAP1 (0.38) HPGDCYP1A2HSD17B10
SCHEMBL16386458 0.67 TGFBR1 (0.38) KDM4ETGFBR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018013430-A2 HETEROCYCLIC COMPOUNDS FOR THE TREATMENT OF ARENAVIRUS INFECTION ARISAN THERAPEUTICS INC. (US) 2018-01-18 WO disclosed