SCHEMBL19831065

SCHEMBL19831065

CCOC(=O)c1c(C(=O)c2ccc(OC)cc2)c2ccc(F)cc2n1-c1ccc(F)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK8 P45983 2/20 0.47
PPARG P37231 1/20 0.46
P2RX3 P56373 3/20 0.45
MAPT P10636 3/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
CCR3 P51677 1/20 0.43
TP53 P04637 2/20 0.43
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
PDE4D Q08499 1/20 0.42
HPGD P15428 2/20 0.41
HTT P42858 2/20 0.41
AKR1C3 P42330 1/20 0.41
AKR1C2 P52895 1/20 0.41
PKM P14618 1/20 0.41
ALOX15 P16050 1/20 0.41
TSHR P16473 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19831224 0.87 MAPK8 (0.48) MAPK8PPARGTP53MEN1KMT2A
SCHEMBL19831040 0.85 MAPK8 (0.52) MAPK8PPARGP2RX3MAPTCYP1A2
SCHEMBL19831199 0.81 CCR3 (0.44) MAPK8CCR3HPGDHTTAKR1C3
SCHEMBL19831197 0.81 ALDH1A1 (0.46) MAPK8MAPTCCR3TP53MEN1
SCHEMBL19831098 0.78 ELANE (0.45) MAPK8MAPTCYP1A2CYP2C9CYP2C19
SCHEMBL19831032 0.78 MAPK1 (0.52) MAPK8HPGDHTTALOX15TSHR
SCHEMBL19831099 0.75 ELANE (0.48) MAPK8PPARGMAPTTP53MEN1
SCHEMBL19831072 0.74 MAPK1 (0.48) MAPK8MAPTKMT2AHPGDHTT
SCHEMBL19831067 0.74 ALOX15 (0.53) MAPTMEN1KMT2AHPGDHTT
SCHEMBL10095274 0.73 TP53 (0.55) PPARGMAPTCYP1A2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018021762-A1 NOVEL COMPOUND, PREPARATION METHOD THEREFOR, AND PHARMACEUTICAL COMPOSITION CONTAINING SAME 현대약품 주식회사 2018-02-01 WO disclosed