SCHEMBL19860036

SCHEMBL19860036

NC(CC(=O)Nc1ccc2cnccc2c1)C(=O)Nc1ccccc1

nearest known ligand 0.66

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 15/20 0.66
ROCK1 Q13464 2/20 0.66
IMPDH2 P12268 2/20 0.64
NOTUM Q6P988 2/20 0.53
SLC1A3 P43003 1/20 0.52
SLC1A2 P43004 1/20 0.52
SLC1A1 P43005 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19860039 0.87 ROCK2 (0.65) ROCK2ROCK1IMPDH2NOTUM
SCHEMBL19860038 0.87 PRMT3 (0.60) ROCK2ROCK1IMPDH2NOTUM
SCHEMBL19860041 0.87 ROCK2 (0.59) ROCK2ROCK1IMPDH2NOTUMSLC1A3
SCHEMBL20353584 0.84 ROCK2 (0.62) ROCK2ROCK1
SCHEMBL20353450 0.84 ROCK2 (0.69) ROCK2ROCK1IMPDH2
SCHEMBL12042256 0.83 ROCK2 (0.55) ROCK2ROCK1IMPDH2NOTUM
SCHEMBL19860037 0.81 NOTUM (0.55) ROCK2ROCK1IMPDH2NOTUM
SCHEMBL20353447 0.81 ROCK2 (0.60) ROCK2ROCK1
SCHEMBL11975549 0.81 ROCK2 (0.57) ROCK2ROCK1IMPDH2NOTUM
SCHEMBL13764336 0.80 ROCK2 (1.00) ROCK2ROCK1IMPDH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9890123-B2 6-aminoisoquinoline compounds AERIE PHARMACEUTICALS, INC. (US) 2018-02-13 US disclosed