SCHEMBL19860039

SCHEMBL19860039

COc1cccc(NC(=O)C(N)CC(=O)Nc2ccc3cnccc3c2)c1

nearest known ligand 0.65

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 15/20 0.65
NOTUM Q6P988 4/20 0.55
ROCK1 Q13464 2/20 0.53
IMPDH2 P12268 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19860036 0.87 ROCK2 (0.66) ROCK2NOTUMROCK1IMPDH2
SCHEMBL19860038 0.84 PRMT3 (0.60) ROCK2NOTUMROCK1IMPDH2
SCHEMBL20353447 0.83 ROCK2 (0.60) ROCK2ROCK1
SCHEMBL19860037 0.83 NOTUM (0.55) ROCK2NOTUMROCK1IMPDH2
SCHEMBL3590824 0.82 NOTUM (0.60) ROCK2NOTUMIMPDH2
SCHEMBL12042256 0.81 ROCK2 (0.55) ROCK2NOTUMROCK1IMPDH2
SCHEMBL19860041 0.79 ROCK2 (0.59) ROCK2NOTUMROCK1IMPDH2
SCHEMBL20353584 0.79 ROCK2 (0.62) ROCK2ROCK1
SCHEMBL20353446 0.79 ROCK2 (0.67) ROCK2ROCK1
SCHEMBL14124407 0.79 ROCK2 (0.66) ROCK2NOTUMROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9890123-B2 6-aminoisoquinoline compounds AERIE PHARMACEUTICALS, INC. (US) 2018-02-13 US disclosed