SCHEMBL19860038

SCHEMBL19860038

CNC(=O)C(N)CC(=O)Nc1ccc2cnccc2c1

nearest known ligand 0.60

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PRMT3 O60678 1/20 0.60
ROCK2 O75116 14/20 0.57
ROCK1 Q13464 2/20 0.57
IMPDH2 P12268 3/20 0.53
NOTUM Q6P988 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12042256 0.89 ROCK2 (0.55) PRMT3ROCK2ROCK1IMPDH2NOTUM
SCHEMBL19860041 0.88 ROCK2 (0.59) PRMT3ROCK2ROCK1IMPDH2NOTUM
SCHEMBL19860036 0.87 ROCK2 (0.66) ROCK2ROCK1IMPDH2NOTUM
SCHEMBL19860037 0.87 NOTUM (0.55) PRMT3ROCK2ROCK1IMPDH2NOTUM
SCHEMBL11975549 0.86 ROCK2 (0.57) PRMT3ROCK2ROCK1IMPDH2NOTUM
SCHEMBL19860039 0.84 ROCK2 (0.65) ROCK2ROCK1IMPDH2NOTUM
SCHEMBL14147299 0.83 RAB9A (0.68) PRMT3ROCK2ROCK1IMPDH2NOTUM
SCHEMBL20353584 0.82 ROCK2 (0.62) ROCK2ROCK1
SCHEMBL20353447 0.82 ROCK2 (0.60) ROCK2ROCK1
SCHEMBL20353452 0.79 ROCK2 (0.68) ROCK2ROCK1IMPDH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9890123-B2 6-aminoisoquinoline compounds AERIE PHARMACEUTICALS, INC. (US) 2018-02-13 US disclosed