SCHEMBL19860041

SCHEMBL19860041

NC(CC(=O)Nc1ccc2cnccc2c1)C(=O)O

nearest known ligand 0.59

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 7/20 0.59
ROCK1 Q13464 3/20 0.59
SLC1A3 P43003 3/20 0.57
SLC1A2 P43004 3/20 0.57
SLC1A1 P43005 3/20 0.57
IMPDH2 P12268 3/20 0.56
PRMT3 O60678 2/20 0.53
NOTUM Q6P988 4/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12042256 0.89 ROCK2 (0.55) ROCK2ROCK1IMPDH2PRMT3NOTUM
SCHEMBL19860038 0.88 PRMT3 (0.60) ROCK2ROCK1IMPDH2PRMT3NOTUM
SCHEMBL19860036 0.87 ROCK2 (0.66) ROCK2ROCK1SLC1A3SLC1A2SLC1A1
SCHEMBL19860037 0.86 NOTUM (0.55) ROCK2ROCK1IMPDH2PRMT3NOTUM
SCHEMBL11975549 0.86 ROCK2 (0.57) ROCK2ROCK1IMPDH2PRMT3NOTUM
SCHEMBL14147299 0.83 RAB9A (0.68) ROCK2ROCK1IMPDH2PRMT3NOTUM
SCHEMBL19859923 0.82 SLC1A3 (0.80) SLC1A3SLC1A2SLC1A1
SCHEMBL12201759 0.81 IMPDH2 (0.61) ROCK2ROCK1IMPDH2PRMT3NOTUM
Hydrochloric Acid SCHEMBL2162309 0.80 IMPDH2 (0.59) ROCK2ROCK1IMPDH2PRMT3NOTUM
Hydrochloric Acid SCHEMBL3564762 0.80 IMPDH2 (0.59) ROCK2ROCK1IMPDH2PRMT3NOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9890123-B2 6-aminoisoquinoline compounds AERIE PHARMACEUTICALS, INC. (US) 2018-02-13 US disclosed