SCHEMBL19860037

SCHEMBL19860037

COC(=O)C(N)CC(=O)Nc1ccc2cnccc2c1

nearest known ligand 0.55

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 5/20 0.55
ROCK2 O75116 11/20 0.54
PRMT3 O60678 2/20 0.53
ROCK1 Q13464 2/20 0.53
IMPDH2 P12268 2/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12042256 0.88 ROCK2 (0.55) NOTUMROCK2PRMT3ROCK1IMPDH2
SCHEMBL19860038 0.87 PRMT3 (0.60) NOTUMROCK2PRMT3ROCK1IMPDH2
SCHEMBL19860041 0.86 ROCK2 (0.59) NOTUMROCK2PRMT3ROCK1IMPDH2
SCHEMBL11975549 0.85 ROCK2 (0.57) NOTUMROCK2PRMT3ROCK1IMPDH2
SCHEMBL19859922 0.84 RAB9A (0.66)
SCHEMBL19860039 0.83 ROCK2 (0.65) NOTUMROCK2ROCK1IMPDH2
SCHEMBL14147299 0.82 RAB9A (0.68) NOTUMROCK2PRMT3ROCK1IMPDH2
SCHEMBL19860036 0.81 ROCK2 (0.66) NOTUMROCK2ROCK1IMPDH2
SCHEMBL20353447 0.81 ROCK2 (0.60) ROCK2ROCK1
SCHEMBL19860094 0.80 NOTUM (0.68) NOTUMROCK2PRMT3ROCK1IMPDH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9890123-B2 6-aminoisoquinoline compounds AERIE PHARMACEUTICALS, INC. (US) 2018-02-13 US disclosed