SCHEMBL19860107

SCHEMBL19860107

O=C(CNCc1cccc(C(F)(F)F)c1)Nc1ccc2cnccc2c1

nearest known ligand 0.57

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 3/20 0.57
TRPV1 Q8NER1 4/20 0.52
IMPDH2 P12268 3/20 0.52
NOTUM Q6P988 4/20 0.48
PRMT3 O60678 2/20 0.47
OPRM1 P35372 1/20 0.47
MEN1 O00255 1/20 0.46
MAPT P10636 1/20 0.46
KMT2A Q03164 1/20 0.46
ROCK1 Q13464 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19860091 0.86 ROCK2 (0.60) ROCK2TRPV1IMPDH2NOTUMPRMT3
SCHEMBL14124375 0.86 ROCK1 (0.59) ROCK2IMPDH2NOTUMPRMT3ROCK1
SCHEMBL14124406 0.86 KDM5A (0.52) ROCK2IMPDH2NOTUMPRMT3ROCK1
SCHEMBL2162616 0.85 IMPDH2 (0.70) ROCK2IMPDH2NOTUMPRMT3MAPT
SCHEMBL2163047 0.84 NOTUM (0.65) ROCK2IMPDH2NOTUMPRMT3ROCK1
SCHEMBL19860110 0.84 IMPDH2 (0.59) ROCK2IMPDH2NOTUMPRMT3ROCK1
SCHEMBL2162395 0.82 ROCK2 (0.61) ROCK2IMPDH2NOTUMPRMT3MEN1
SCHEMBL19860124 0.82 IMPDH2 (0.59) IMPDH2NOTUMPRMT3
SCHEMBL14124373 0.81 NOTUM (0.55) ROCK2IMPDH2NOTUMPRMT3MAPT
SCHEMBL19860040 0.81 PRMT3 (0.53) ROCK2IMPDH2NOTUMPRMT3ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9890123-B2 6-aminoisoquinoline compounds AERIE PHARMACEUTICALS, INC. (US) 2018-02-13 US disclosed