SCHEMBL19860124

SCHEMBL19860124

O=C(CNCc1ccncc1)Nc1ccc2cnccc2c1

nearest known ligand 0.59

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
IMPDH2 P12268 3/20 0.59
PRMT3 O60678 12/20 0.56
KDM4E B2RXH2 1/20 0.54
ALDH1A1 P00352 1/20 0.54
NOTUM Q6P988 4/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2162616 0.93 IMPDH2 (0.70) IMPDH2PRMT3KDM4EALDH1A1NOTUM
SCHEMBL19860106 0.90 ROCK1 (0.57) IMPDH2PRMT3NOTUM
SCHEMBL19860110 0.89 IMPDH2 (0.59) IMPDH2PRMT3NOTUM
SCHEMBL19860042 0.88 MEN1 (0.60) IMPDH2PRMT3KDM4EALDH1A1NOTUM
SCHEMBL14124377 0.86 PRMT3 (0.51) IMPDH2PRMT3KDM4EALDH1A1NOTUM
SCHEMBL14136014 0.86 LMNA (0.67) IMPDH2PRMT3KDM4EALDH1A1NOTUM
SCHEMBL19860109 0.86 PRMT3 (0.50) IMPDH2PRMT3NOTUM
SCHEMBL14124375 0.85 ROCK1 (0.59) IMPDH2PRMT3NOTUM
SCHEMBL2163047 0.85 NOTUM (0.65) IMPDH2PRMT3NOTUM
SCHEMBL19860105 0.84 PRMT3 (0.62) IMPDH2PRMT3NOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9890123-B2 6-aminoisoquinoline compounds AERIE PHARMACEUTICALS, INC. (US) 2018-02-13 US disclosed