SCHEMBL19860091

SCHEMBL19860091

O=C(CCc1cccc(C(F)(F)F)c1)Nc1ccc2cnccc2c1

nearest known ligand 0.60

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 4/20 0.60
TRPV1 Q8NER1 3/20 0.54
PRMT3 O60678 1/20 0.53
IMPDH2 P12268 2/20 0.52
MCHR1 Q99705 3/20 0.52
NOTUM Q6P988 4/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2164396 0.89 IMPDH2 (0.58) ROCK2TRPV1PRMT3IMPDH2MCHR1
SCHEMBL19860107 0.86 ROCK2 (0.57) ROCK2TRPV1PRMT3IMPDH2NOTUM
SCHEMBL3566775 0.84 PRMT3 (0.72) ROCK2PRMT3IMPDH2NOTUM
SCHEMBL2164137 0.82 PRMT3 (0.69) ROCK2PRMT3IMPDH2NOTUM
SCHEMBL19860067 0.81 PRMT3 (0.54) ROCK2PRMT3IMPDH2NOTUM
SCHEMBL19860079 0.80 ALDH1A1 (0.61) ROCK2PRMT3IMPDH2NOTUM
SCHEMBL19860089 0.80 ROCK2 (0.55) ROCK2PRMT3IMPDH2NOTUM
SCHEMBL19860064 0.80 PRMT3 (0.54) ROCK2PRMT3IMPDH2NOTUM
SCHEMBL19860062 0.80 ALDH1A1 (0.61) ROCK2PRMT3IMPDH2NOTUM
SCHEMBL19860082 0.79 ROCK1 (0.60) ROCK2PRMT3IMPDH2MCHR1NOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9890123-B2 6-aminoisoquinoline compounds AERIE PHARMACEUTICALS, INC. (US) 2018-02-13 US disclosed