SCHEMBL19924765

SCHEMBL19924765

O=C(NC(Cc1cccc(C(F)(F)F)n1)C(=O)O)OCc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 8/20 0.47
ITGA2B P08514 8/20 0.47
ALDH1A1 P00352 1/20 0.47
ALOX15 P16050 1/20 0.47
TACR1 P25103 2/20 0.46
CTSL P07711 2/20 0.45
CTSS P25774 2/20 0.45
CTSB P07858 1/20 0.45
CTSK P43235 1/20 0.45
CTRB1 P17538 2/20 0.44
CASP1 P29466 1/20 0.44
PPARG P37231 1/20 0.44
PPARA Q07869 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19924764 1.00 ITGB3 (0.47) ITGB3ITGA2BALDH1A1ALOX15TACR1
SCHEMBL19924784 0.91 ALDH1A1 (0.53) ALDH1A1ALOX15TACR1CTSLCTSS
SCHEMBL19924783 0.91 ALDH1A1 (0.53) ALDH1A1ALOX15TACR1CTSLCTSS
SCHEMBL7452849 0.79 CTSL (0.58) ITGB3ITGA2BALDH1A1TACR1CTSL
SCHEMBL1795688 0.78 TGM2 (0.60) ITGB3ITGA2BTACR1CTSLCTSS
SCHEMBL4368353 0.78 FPR2 (0.62) ITGB3ITGA2BALDH1A1ALOX15TACR1
SCHEMBL3987614 0.78 FPR2 (0.62) ITGB3ITGA2BALDH1A1ALOX15TACR1
SCHEMBL220648 0.78 TACR1 (0.68) ITGB3ITGA2BALDH1A1ALOX15TACR1
SCHEMBL7372270 0.78 TACR1 (0.68) ITGB3ITGA2BALDH1A1ALOX15TACR1
SCHEMBL479010 0.78 TACR1 (0.68) ITGB3ITGA2BALDH1A1ALOX15TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018042343-A2 COMPOUNDS THAT INHIBIT 3C AND 3CL PROTEASES AND METHODS OF USE THEREOF GLAXOSMITHKLINE INTELLECTUAL PROPERTY (NO.2) LIMITED (GB) 2018-03-08 WO disclosed