SCHEMBL19933674

SCHEMBL19933674

c1ccc(-c2nc(-c3ccccc3)nc(-c3ccc(-n4c5ccccc5c5cc(-c6ccc7oc8cccc(-c9nc(-c%10ccccc%10)nc(-c%10ccccc%10)n9)c8c7c6)ccc54)cc3)n2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 3/20 0.35
KDM4E B2RXH2 2/20 0.35
ATM Q13315 2/20 0.35
PLA2G2A P14555 3/20 0.35
PLA2G4A P47712 3/20 0.35
PLA2G10 O15496 1/20 0.35
PTGER4 P35408 1/20 0.33
SIRT2 Q8IXJ6 1/20 0.32
SIRT1 Q96EB6 1/20 0.32
PIM1 P11309 1/20 0.31
CSNK2A2 P19784 1/20 0.31
CSNK2B P67870 1/20 0.31
PIM3 Q86V86 1/20 0.31
PIM2 Q9P1W9 1/20 0.31
CHEK2 O96017 1/20 0.31
ALDH1A1 P00352 3/20 0.31
HPGD P15428 3/20 0.31
TSHR P16473 2/20 0.31
RAC2 P15153 1/20 0.31
RAC3 P60763 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25944400 0.99 PLA2G2A (0.36) L3MBTL1KDM4EATMPLA2G2APLA2G4A
SCHEMBL22145856 0.99 PLA2G2A (0.36) L3MBTL1KDM4EATMPLA2G2APLA2G4A
SCHEMBL17252528 0.99 PLA2G2A (0.36) L3MBTL1KDM4EATMPLA2G2APLA2G4A
SCHEMBL23559222 0.98 KDM4E (0.38) L3MBTL1KDM4EATMPLA2G2APLA2G4A
SCHEMBL17252634 0.98 KDM4E (0.38) L3MBTL1KDM4EATMPLA2G2APLA2G4A
SCHEMBL17252747 0.98 KDM4E (0.38) L3MBTL1KDM4EATMPLA2G2APLA2G4A
SCHEMBL29353592 0.98 KDM4E (0.38) L3MBTL1KDM4EATMPLA2G2APLA2G4A
SCHEMBL22257773 0.97 PLA2G2A (0.35) L3MBTL1KDM4EATMPLA2G2APLA2G4A
SCHEMBL22257568 0.97 PLA2G2A (0.35) L3MBTL1KDM4EATMPLA2G2APLA2G4A
SCHEMBL22022426 0.97 KDM4E (0.36) L3MBTL1KDM4EATMPLA2G2APLA2G4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 43 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11917903-B2 Metal complexes UDC IRELAND LIMITED (IE) 2024-02-27 US disclosed
US-11917903-B2 Metal complexes UDC IRELAND LIMITED (IE) 2024-02-27 US disclosed
US-11877511-B2 Materials for organic light emitting devices MERCK PATENT GMBH (DE) 2024-01-16 US disclosed
US-11877511-B2 Materials for organic light emitting devices MERCK PATENT GMBH (DE) 2024-01-16 US disclosed
US-20230320191-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2023-10-05 US disclosed
US-20230320191-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2023-10-05 US disclosed
US-20230292596-A1 MATERIALS FOR ORGANIC ELECTROLUMINESCENT DEVICES MERCK PATENT GMBH (DE) 2023-09-14 US disclosed
US-20230292596-A1 MATERIALS FOR ORGANIC ELECTROLUMINESCENT DEVICES MERCK PATENT GMBH (DE) 2023-09-14 US disclosed
US-20230271989-A1 METAL COMPLEXES UDC IRELAND LIMITED (IE) 2023-08-31 US disclosed
US-20230271989-A1 METAL COMPLEXES UDC IRELAND LIMITED (IE) 2023-08-31 US disclosed
US-20200251660-A1 MATERIALS FOR ORGANIC LIGHT EMITTING DEVICES MERCK PATENT GMBH (DE) 2020-08-06 US disclosed
US-20200207794-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2020-07-02 US disclosed
US-20200052213-A1 BINUCLEAR METAL COMPLEXES AND ELECTRONIC DEVICES, IN PARTICULAR ORGANIC ELECTROLUMINESCENT DEVICES CONTAINING SAID METAL COMPLEXES MERCK PATENT GMBH (DE) 2020-02-13 US disclosed
US-20190292210-A1 BINUCLEAR METAL COMPLEXES FOR USE AS EMITTERS IN ORGANIC ELECTROLUMINESCENT DEVICES MERCK PATENT GMBH (DE) 2019-09-26 US disclosed
US-20190252628-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2019-08-15 US disclosed
US-20190202851-A1 BINUCLEAR AND TRINUCLEAR METAL COMPLEXES COMPOSED OF TWO INTER-LINKED TRIPODAL HEXADENTATE LIGANDS FOR USE IN ELECTROLUMINESCENT DEVICES MERCK PATENT GMBH (DE) 2019-07-04 US disclosed
WO-2019020538-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2019-01-31 WO disclosed
WO-2018069197-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2018-04-19 WO disclosed
WO-2018054798-A1 BINUCLEAR METAL COMPLEXES FOR USE AS EMITTERS IN ORGANIC ELECTROLUMINESCENT DEVICES MERCK PATENT GMBH (DE) 2018-03-29 WO disclosed
WO-2018041769-A1 BINUCLEAR AND TRINUCLEAR METAL COMPLEXES COMPOSED OF TWO INTER-LINKED TRIPODAL HEXADENTATE LIGANDS FOR USE IN ELECTROLUMINESCENT DEVICES MERCK PATENT GMBH (DE) 2018-03-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (11 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190202851-A1 BINUCLEAR AND TRINUCLEAR METAL COMPLEXES COMPOSED OF TWO INTER-LINKED TRIPODAL HEXADENTATE LIGANDS FOR USE IN ELECTROLUMINESCENT DEVICES PARN, PUF60, PARG L3MBTL1 1520/4885KDM4E 4048/4885ATM 3697/4885
US-20190252628-A1 METAL COMPLEXES AP1M1, AP2M1, AP3M1 L3MBTL1 3031/4885KDM4E 3877/4885ATM 4131/4885
US-20190292210-A1 BINUCLEAR METAL COMPLEXES FOR USE AS EMITTERS IN ORGANIC ELECTROLUMINESCENT DEVICES AP2M1, MCU, AP3M1 L3MBTL1 2504/4885KDM4E 4613/4885ATM 4246/4885
US-20200251660-A1 MATERIALS FOR ORGANIC LIGHT EMITTING DEVICES DDT, ESD, ETFA L3MBTL1 565/4885KDM4E 3065/4885ATM 4454/4885
US-20230320191-A1 METAL COMPLEXES IMMT, MCU, SOD1 L3MBTL1 3259/4885KDM4E 4470/4885ATM 4048/4885
US-20230292596-A1 MATERIALS FOR ORGANIC ELECTROLUMINESCENT DEVICES OR10J3, EPCAM, L1CAM L3MBTL1 1208/4885KDM4E 2021/4885ATM 2990/4885
US-20230271989-A1 METAL COMPLEXES AP3M1, AP1M1, AP2M1 L3MBTL1 2773/4885KDM4E 3576/4885ATM 3098/4885
US-11877511-B2 Materials for organic light emitting devices DDT, ESD, ETFA L3MBTL1 565/4885KDM4E 3065/4885ATM 4454/4885
US-20200207794-A1 METAL COMPLEXES IMMT, MCU, SOD1 L3MBTL1 3259/4885KDM4E 4470/4885ATM 4048/4885
US-20200052213-A1 BINUCLEAR METAL COMPLEXES AND ELECTRONIC DEVICES, IN PARTICULAR ORGANIC ELECTROLUMINESCENT DEVICES CONTAINING SAID METAL COMPLEXES BICRA, NCLN, IMMT L3MBTL1 3344/4885KDM4E 3160/4885ATM 4082/4885
US-11917903-B2 Metal complexes NCLN, BICRA, AP3M1 L3MBTL1 2532/4885KDM4E 3870/4885ATM 3416/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.