SCHEMBL19953095

SCHEMBL19953095

Fc1cc(Cl)ccc1-n1c(-c2c(F)cccc2F)cnc1I

nearest known ligand 0.53

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 3/20 0.38
PDE4D Q08499 3/20 0.38
EGLN2 Q96KS0 1/20 0.36
AOC3 Q16853 5/20 0.35
CYP3A4 P08684 2/20 0.34
SLC22A1 O15245 1/20 0.34
ABCB11 O95342 1/20 0.34
DRD3 P35462 1/20 0.34
OPRK1 P41145 1/20 0.34
SLC22A12 Q96S37 1/20 0.34
PDE2A O00408 1/20 0.33
PDE10A Q9Y233 1/20 0.33
TRPM5 Q9NZQ8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19953169 0.72 CYP3A4 (0.43) EGLN2CYP3A4PDE2APDE10ATRPM5
SCHEMBL1074708 0.68 PTGS2 (0.42) PDE4DAOC3CYP3A4SLC22A1ABCB11
SCHEMBL19953055 0.68 PTGS2 (0.37) EGLN2PDE2APDE10ATRPM5
SCHEMBL24075077 0.63 EGLN2 (0.42) EGLN2
SCHEMBL20575403 0.62 MYC (0.54) AOC3SLC22A12
SCHEMBL23510074 0.62 SLC22A12 (0.45) PDE4BPDE4DAOC3SLC22A12
SCHEMBL30955009 0.61 HDAC4 (0.36)
SCHEMBL19967210 0.59 CCR2 (0.34) CYP3A4SLC22A12PDE2APDE10A
SCHEMBL1110963 0.59 PTGS2 (0.44) AOC3
SCHEMBL19953203 0.58 PTGS2 (0.43) AOC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018048969-A1 MULTI-TARGETED HETEROCYCLIC COMPOUNDS FOR THE TREATMENT OF NEURODEGENERATIVE DISEASES THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2018-03-15 WO disclosed