SCHEMBL19967210

SCHEMBL19967210

Fc1cc(Cl)ccc1N1C(c2c(F)cccc2F)=CNC1Cl

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 2/20 0.34
CCR1 P32246 1/20 0.34
CCR5 P51681 1/20 0.34
SLC22A12 Q96S37 1/20 0.32
PDE2A O00408 1/20 0.30
PDE10A Q9Y233 1/20 0.30
NOTUM Q6P988 1/20 0.30
CYP3A4 P08684 1/20 0.30
MAPT P10636 1/20 0.30
PTGES O14684 1/20 0.30
SLC6A2 P23975 1/20 0.30
SLC6A4 P31645 1/20 0.30
SLC6A3 Q01959 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19953055 0.65 PTGS2 (0.37) PDE2APDE10A
SCHEMBL19953169 0.61 CYP3A4 (0.43) PDE2APDE10ACYP3A4
SCHEMBL11186084 0.59 PPOX (0.46) CCR2CCR1CCR5NOTUM
SCHEMBL19953095 0.59 PDE4B (0.38) SLC22A12PDE2APDE10ACYP3A4
SCHEMBL24628518 0.58 CHRNB2 (0.49)
SCHEMBL19707985 0.58 CA1 (0.43) CCR2CCR1CCR5MAPT
SCHEMBL30273429 0.58 MEN1 (0.53) CYP3A4
SCHEMBL7729256 0.58 MEN1 (0.53) CYP3A4
SCHEMBL30232617 0.57 CHRNB4 (0.44)
SCHEMBL16480401 0.56 NOTUM (0.54) CCR2CCR1CCR5NOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018048969-A1 MULTI-TARGETED HETEROCYCLIC COMPOUNDS FOR THE TREATMENT OF NEURODEGENERATIVE DISEASES THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2018-03-15 WO disclosed