SCHEMBL19953561

SCHEMBL19953561

COC(=O)C1(F)C(=O)N(C)Cc2ccccc21

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 2/20 0.39
OPRK1 P41145 2/20 0.39
OPRL1 P41146 2/20 0.39
BRD4 O60885 1/20 0.39
CREBBP Q92793 1/20 0.39
ALDH1A1 P00352 1/20 0.37
NOTUM Q6P988 1/20 0.36
PARP1 P09874 1/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
POLB P06746 1/20 0.33
IDH1 O75874 1/20 0.33
SCN9A Q15858 1/20 0.33
TAS1R3 Q7RTX0 1/20 0.33
TAS1R1 Q7RTX1 1/20 0.33
TAS1R2 Q8TE23 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19960571 0.79 GRM7 (0.39) OPRM1OPRK1OPRL1MEN1KMT2A
SCHEMBL8705275 0.66 KMT2A (0.47) OPRM1OPRK1OPRL1BRD4CREBBP
SCHEMBL8704499 0.63 OPRM1 (0.39) OPRM1OPRK1OPRL1BRD4CREBBP
SCHEMBL547428 0.63 MEN1 (0.44) ALDH1A1MEN1KMT2APOLB
SCHEMBL14104811 0.63 MEN1 (0.38) OPRM1ALDH1A1NOTUMMEN1KMT2A
SCHEMBL8462462 0.63 KDM4E (0.42) ALDH1A1NOTUMMEN1KMT2APOLB
SCHEMBL15609020 0.62 SIGMAR1 (0.43) ALDH1A1MEN1KMT2A
SCHEMBL22744702 0.62 HTT (0.44) ALDH1A1MEN1KMT2APOLB
SCHEMBL30972513 0.62 MAPT (0.49) ALDH1A1MEN1KMT2A
SCHEMBL1206839 0.61 ALDH1A1 (0.45) ALDH1A1MEN1KMT2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018047983-A1 INDANE DERIVATIVES USEFUL AS MODULATORS OF MGLUR7 TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-03-15 WO disclosed
WO-2018047983-A1 INDANE DERIVATIVES USEFUL AS MODULATORS OF MGLUR7 TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-03-15 WO disclosed