SCHEMBL19960632

SCHEMBL19960632

COC(=O)C1OC(=O)Nc2ccccc21

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.43
CYP2D6 P10635 1/20 0.41
ALDH1A1 P00352 6/20 0.39
KDM4E B2RXH2 4/20 0.39
MAPT P10636 4/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
BACE1 P56817 1/20 0.39
ITGA4 P13612 1/20 0.37
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
IDO1 P14902 1/20 0.36
TDO2 P48775 1/20 0.36
HPGDS O60760 1/20 0.35
HSD17B10 Q99714 2/20 0.35
POLB P06746 1/20 0.35
HPGD P15428 1/20 0.35
HTT P42858 2/20 0.35
NLRP3 Q96P20 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19960649 0.84 EGFR (0.39) EGFRCYP2D6ALDH1A1KDM4EMAPT
SCHEMBL6024348 0.74 EGFR (0.49) EGFRALDH1A1KDM4EMAPTL3MBTL1
SCHEMBL19960702 0.73 FABP5 (0.41) ALDH1A1KDM4EMAPTNPC1RAB9A
SCHEMBL7681777 0.73 MAPT (0.58) EGFRALDH1A1KDM4EMAPTL3MBTL1
SCHEMBL11197568 0.72 PARP1 (0.49) ALDH1A1KDM4EMAPTL3MBTL1IDO1
SCHEMBL10957521 0.72 ALDH1A1 (0.41) EGFRALDH1A1KDM4EMAPTL3MBTL1
SCHEMBL19960475 0.71 EGFR (0.38) EGFRALDH1A1KDM4EMAPTL3MBTL1
SCHEMBL11340291 0.69 EGFR (0.36) EGFRCYP2D6ALDH1A1KDM4EMAPT
SCHEMBL19960622 0.69 HDAC4 (0.44) EGFRCYP2D6ALDH1A1KDM4EMAPT
SCHEMBL11208873 0.68 HTR5A (0.41) ALDH1A1KDM4EMAPTL3MBTL1IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018047983-A1 INDANE DERIVATIVES USEFUL AS MODULATORS OF MGLUR7 TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-03-15 WO disclosed