SCHEMBL19976970

SCHEMBL19976970

COc1cccc(NC(=O)C(C)NC(=O)c2ccccc2)c1C

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.53
RAB9A P51151 3/20 0.53
GPR139 Q6DWJ6 2/20 0.48
ALDH1A1 P00352 2/20 0.46
LMNA P02545 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
MAPT P10636 1/20 0.46
KMT2A Q03164 3/20 0.45
RXFP1 Q9HBX9 1/20 0.45
HPGD P15428 1/20 0.45
HTT P42858 1/20 0.45
LPAR1 Q92633 1/20 0.44
KCNK3 O14649 1/20 0.44
KCNK9 Q9NPC2 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
MEN1 O00255 2/20 0.44
HDAC1 Q13547 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19976980 0.90 NPC1 (0.66) NPC1RAB9AALDH1A1LMNATDP1
SCHEMBL19977134 0.89 HDAC1 (0.46) NPC1RAB9AGPR139LMNAKMT2A
SCHEMBL19976955 0.84 POLB (0.53) NPC1RAB9AALDH1A1LMNAMAPT
SCHEMBL19976954 0.83 KMT2A (0.53) NPC1RAB9AALDH1A1LMNATDP1
SCHEMBL16999305 0.82 USP30 (0.55) GPR139HDAC1
SCHEMBL19977072 0.82 LMNA (0.54) GPR139LMNAKMT2AHPGDHTT
SCHEMBL19977018 0.82 SMN1; SMN2 (0.50) NPC1RAB9AALDH1A1LMNAKMT2A
SCHEMBL19976952 0.81 APLNR (0.57) NPC1RAB9AALDH1A1LMNAMAPT
SCHEMBL19977070 0.81 KCNK3 (0.48) RAB9AALDH1A1LMNAMAPTHPGD
SCHEMBL19976971 0.81 HDAC1 (0.53) NPC1RAB9ALMNAKMT2ARXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9919998-B2 Antibacterial agents: Nα-aroyl-N-aryl-phenylalaninamides RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2018-03-20 US disclosed