SCHEMBL19976995

SCHEMBL19976995

Cc1ccccc1C(=O)NC(C)C(=O)Nc1cc(Cl)ccc1N1CCNCC1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.48
KDM4E B2RXH2 4/20 0.48
NPSR1 Q6W5P4 3/20 0.48
HPGD P15428 3/20 0.48
TSHR P16473 2/20 0.48
POLB P06746 1/20 0.48
HSD17B10 Q99714 1/20 0.48
KCNMA1 Q12791 1/20 0.46
IDH2 P48735 1/20 0.46
L3MBTL1 Q9Y468 2/20 0.44
ATM Q13315 1/20 0.44
BACE1 P56817 2/20 0.44
MAPT P10636 3/20 0.43
BRPF1 P55201 2/20 0.43
GAA P10253 2/20 0.43
LMNA P02545 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
CRHBP P24387 1/20 0.43
HTT P42858 1/20 0.43
CRHR2 Q13324 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19977001 0.90 KMT2A (0.47) ALDH1A1KDM4ENPSR1HPGDTSHR
SCHEMBL19977130 0.89 L3MBTL1 (0.44) ALDH1A1KDM4EL3MBTL1ATMBACE1
SCHEMBL19976964 0.88 L3MBTL1 (0.58) ALDH1A1NPSR1TSHRPOLBHSD17B10
SCHEMBL16993937 0.86 CTSV (0.51) ALDH1A1KDM4ENPSR1HPGDTSHR
SCHEMBL19976968 0.81 KCNMA1 (0.57) ALDH1A1KDM4ENPSR1HPGDPOLB
SCHEMBL19977012 0.80 ALDH1A1 (0.46) ALDH1A1KDM4ENPSR1HPGDTSHR
SCHEMBL19977068 0.78 BACE1 (0.57) ALDH1A1KDM4ENPSR1HPGDTSHR
SCHEMBL19977110 0.78 BACE1 (0.48) ALDH1A1NPSR1HPGDPOLBBACE1
SCHEMBL19977098 0.77 KDM4E (0.51) ALDH1A1KDM4ENPSR1HPGDTSHR
SCHEMBL19977129 0.77 ALDH1A1 (0.57) ALDH1A1NPSR1TSHRPOLBHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3102193-B1 ANTIBACTERIAL AGENTS: N(ALPHA)-AROYL-N-ARYL-PHENYLALANINAMIDES UNIV RUTGERS (US) 2023-01-11 EP disclosed
US-9919998-B2 Antibacterial agents: Nα-aroyl-N-aryl-phenylalaninamides RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2018-03-20 US disclosed