SCHEMBL19977033

SCHEMBL19977033

CC(NC(=O)c1ccccc1Cl)C(=O)Nc1cccc2cc[nH]c12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
GRM5 P41594 1/20 0.44
PYGL P06737 1/20 0.43
CYP1A2 P05177 1/20 0.43
HPGD P15428 1/20 0.43
CYP2C19 P33261 1/20 0.43
KDR P35968 1/20 0.42
KMT2A Q03164 1/20 0.41
HTT P42858 2/20 0.41
AHR P35869 1/20 0.40
CCKAR P32238 1/20 0.40
ROCK2 O75116 1/20 0.40
KEAP1 Q14145 1/20 0.40
KDM4E B2RXH2 1/20 0.40
NR3C1 P04150 1/20 0.40
PGR P06401 1/20 0.40
NR3C2 P08235 1/20 0.40
AR P10275 1/20 0.40
PDPK1 O15530 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19977034 0.88 PARP1 (0.46) TRPV1GRM5PYGLHPGDKMT2A
SCHEMBL19976949 0.87 KMT2A (0.45) TRPV1SMN1; SMN2GRM5KMT2AHTT
SCHEMBL19976902 0.84 SMN1; SMN2 (0.45) TRPV1SMN1; SMN2CYP1A2CYP2C19KMT2A
SCHEMBL16993985 0.82 PSMB5 (0.46) PYGLCCKARROCK2
SCHEMBL19976910 0.78 PGR (0.52) SMN1; SMN2PYGLCYP1A2HPGDCYP2C19
SCHEMBL19976903 0.78 MEN1 (0.50) TRPV1HPGDKMT2ANR3C1PGR
SCHEMBL19977127 0.76 TRPV1 (0.54) TRPV1KMT2AHTT
SCHEMBL19977030 0.75 MAPT (0.57) SMN1; SMN2PYGLKMT2AHTTKDM4E
SCHEMBL19977046 0.73 KMT2A (0.50) SMN1; SMN2PYGLCYP1A2HPGDCYP2C19
SCHEMBL19976933 0.72 PABPC1 (0.73) SMN1; SMN2KDRKMT2AHTTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9919998-B2 Antibacterial agents: Nα-aroyl-N-aryl-phenylalaninamides RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2018-03-20 US disclosed