SCHEMBL19976949

SCHEMBL19976949

CC(NC(=O)c1ccccc1F)C(=O)Nc1cccc2cc[nH]c12

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.45
MEN1 O00255 2/20 0.45
HTT P42858 3/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
LMNA P02545 1/20 0.41
TRPV1 Q8NER1 1/20 0.41
POLB P06746 1/20 0.40
CCKAR P32238 1/20 0.40
HDAC3 O15379 1/20 0.40
HDAC1 Q13547 1/20 0.40
KEAP1 Q14145 1/20 0.40
KDM4E B2RXH2 1/20 0.40
NR3C1 P04150 1/20 0.40
PGR P06401 1/20 0.40
NR3C2 P08235 1/20 0.40
AR P10275 1/20 0.40
PDPK1 O15530 1/20 0.39
GRM5 P41594 1/20 0.39
GAA P10253 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19977034 0.88 PARP1 (0.46) KMT2AMEN1HTTLMNATRPV1
SCHEMBL19977033 0.87 TRPV1 (0.45) KMT2AHTTSMN1; SMN2TRPV1CCKAR
SCHEMBL19976902 0.84 SMN1; SMN2 (0.45) KMT2AMEN1SMN1; SMN2LMNATRPV1
SCHEMBL19977090 0.82 DHPS (0.46) KMT2AMEN1HTTSMN1; SMN2LMNA
SCHEMBL16994055 0.82 CTSL (0.47) KMT2AMEN1CCKAR
SCHEMBL19977103 0.81 KMT2A (0.46) KMT2AMEN1HTTSMN1; SMN2LMNA
SCHEMBL19976906 0.78 PGR (0.52) KMT2AMEN1HTTSMN1; SMN2LMNA
SCHEMBL19976903 0.78 MEN1 (0.50) KMT2AMEN1TRPV1POLBNR3C1
SCHEMBL19977029 0.76 KDM4E (0.54) KMT2AMEN1HTTLMNATRPV1
SCHEMBL19976990 0.75 KMT2A (0.60) KMT2AMEN1HTTSMN1; SMN2HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9919998-B2 Antibacterial agents: Nα-aroyl-N-aryl-phenylalaninamides RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2018-03-20 US disclosed