SCHEMBL19977034

SCHEMBL19977034

Cc1ccccc1C(=O)NC(C)C(=O)Nc1cccc2cc[nH]c12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.46
LMNA P02545 3/20 0.42
MEN1 O00255 1/20 0.42
ALOX12 P18054 1/20 0.42
KMT2A Q03164 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
PYGL P06737 1/20 0.41
CCKAR P32238 1/20 0.41
KEAP1 Q14145 1/20 0.41
PGR P06401 2/20 0.40
HTT P42858 2/20 0.40
NR3C1 P04150 1/20 0.40
NR3C2 P08235 1/20 0.40
AR P10275 1/20 0.40
KDM4E B2RXH2 1/20 0.40
SCN1A P35498 1/20 0.40
SCN2A Q99250 1/20 0.40
SCN3A Q9NY46 1/20 0.40
PDPK1 O15530 1/20 0.40
GRM5 P41594 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19976949 0.88 KMT2A (0.45) LMNAMEN1KMT2ACCKARKEAP1
SCHEMBL19977033 0.88 TRPV1 (0.45) KMT2APYGLCCKARKEAP1PGR
SCHEMBL19976902 0.85 SMN1; SMN2 (0.45) PARP1LMNAMEN1KMT2ACCKAR
SCHEMBL16994027 0.83 CTSV (0.48) MEN1KMT2APYGLCCKAR
SCHEMBL19976994 0.81 PGR (0.57) LMNAMEN1ALOX12KMT2ANPSR1
SCHEMBL19976997 0.80 MAPT (0.41) PARP1LMNAMEN1ALOX12KMT2A
SCHEMBL19976903 0.79 MEN1 (0.50) PARP1MEN1KMT2ANPSR1PGR
SCHEMBL19977084 0.77 DHPS (0.46) PARP1LMNAMEN1ALOX12KMT2A
SCHEMBL19976940 0.76 TRPV1 (0.55) LMNAMEN1KMT2AHTTMAPT
SCHEMBL19977032 0.75 MAPT (0.55) MEN1ALOX12KMT2ANPSR1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9919998-B2 Antibacterial agents: Nα-aroyl-N-aryl-phenylalaninamides RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2018-03-20 US disclosed