SCHEMBL19981909

SCHEMBL19981909

CCNCCNc1ccc(N)nc1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 3/20 0.40
ADRA2B P18089 3/20 0.40
ADRA2C P18825 3/20 0.40
MAPT P10636 3/20 0.39
NOS3 P29474 1/20 0.38
NOS2 P35228 1/20 0.38
GAA P10253 2/20 0.36
RRM2 P31350 3/20 0.36
BRAF P15056 1/20 0.34
NAMPT P43490 1/20 0.33
ALPL P05186 1/20 0.33
STK17A Q9UEE5 1/20 0.33
ROCK1 Q13464 1/20 0.33
ILK Q13418 1/20 0.32
NSD2 O96028 1/20 0.32
KMT2A Q03164 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
PIK3CA P42336 1/20 0.32
MTOR P42345 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2487033 0.83 ADRA2A (0.53) ADRA2AADRA2BADRA2CMAPTNOS3
SCHEMBL20929322 0.82 MAPT (0.42) ADRA2AADRA2BADRA2CMAPTNOS3
SCHEMBL5694416 0.82 MAOA (0.43) MAPTNOS3NOS2GAANAMPT
SCHEMBL12102026 0.80 MAPT (0.46) ADRA2AADRA2BADRA2CMAPTGAA
SCHEMBL22175094 0.78 MAPT (0.38) ADRA2AADRA2BADRA2CMAPTNOS3
SCHEMBL18779716 0.77 KCNH3 (0.40) ADRA2AADRA2BADRA2CNOS3NOS2
SCHEMBL28820864 0.76 NOS3 (0.42) ADRA2AADRA2BADRA2CMAPTNOS3
SCHEMBL16963191 0.76 HRH3 (0.47) NOS3NOS2GAA
SCHEMBL2483964 0.76 KCNH3 (0.48) MAPTNOS3NOS2GAAALPL
SCHEMBL20878669 0.76 MTNR1A (0.48) NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2365970-B1 PYRIDAZINONES AND THEIR USE AS BTK INHIBITORS GILEAD CONNECTICUT INC (US) 2018-03-21 EP disclosed