SCHEMBL19984846

SCHEMBL19984846

COc1ccccc1-c1nnc([C@H](C)NC(=O)c2cccc(C(=O)O)c2)o1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARD Q03181 2/20 0.49
NPSR1 Q6W5P4 1/20 0.47
HSD17B10 Q99714 1/20 0.47
NPC1 O15118 3/20 0.45
RAB9A P51151 3/20 0.45
KDM4E B2RXH2 3/20 0.45
MAPT P10636 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
LMNA P02545 2/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
ALDH1A1 P00352 4/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
KMT2A Q03164 1/20 0.44
HPGD P15428 2/20 0.43
GAA P10253 1/20 0.43
PKM P14618 1/20 0.43
TP53 P04637 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19984823 0.86 ADAMTS4 (0.55) PPARDNPC1RAB9AKDM4EMAPT
SCHEMBL19984825 0.82 ADAMTS4 (0.57) PPARDNPC1RAB9AKDM4EMAPT
SCHEMBL19984976 0.79 APLNR (0.54) PPARDMAPTKMT2AHPGDGAA
SCHEMBL19984967 0.79 ADAMTS4 (0.54) PPARDNPC1RAB9AKDM4EMAPT
SCHEMBL12171886 0.78 PPARD (0.56) PPARDHSD17B10NPC1RAB9AKDM4E
SCHEMBL19984971 0.76 ADAMTS4 (0.45) PPARDNPC1RAB9AKDM4ESMN1; SMN2
SCHEMBL19984985 0.76 ADAMTS4 (0.55) HPGDGAA
SCHEMBL2435361 0.74 PPARD (0.50) PPARDHSD17B10NPC1RAB9AKDM4E
SCHEMBL12171732 0.71 NPC1 (0.66) PPARDNPC1RAB9AKDM4EMAPT
SCHEMBL11615095 0.70 ALDH1A1 (0.58) HSD17B10NPC1RAB9AKDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018051255-A1 CYCLIC SUBSTITUTED-1,3,4-OXADIAZOLE AND THIADIAZOLE COMPOUNDS AS IMMUNOMODULATORS AURIGENE DISCOVERY TECHNOLOGIES LIMITED (IN) 2018-03-22 WO disclosed