SCHEMBL1999222

SCHEMBL1999222

O=C(c1cnc(-c2ccccn2)o1)c1c(Cl)n(Cc2ccc(Cl)cc2)c2ccc(O)cc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.40
PKM P14618 3/20 0.40
GAA P10253 2/20 0.40
ALDH1A1 P00352 2/20 0.40
S1PR3 Q99500 3/20 0.39
KDM4E B2RXH2 2/20 0.39
LMNA P02545 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
ALOX5AP P20292 3/20 0.37
CYP3A4 P08684 2/20 0.37
CYP2C9 P11712 2/20 0.37
ALOX5 P09917 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C19 P33261 1/20 0.36
MAPK10 P53779 1/20 0.36
CNR1 P21554 1/20 0.36
CNR2 P34972 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2007882 0.94 HSD17B10 (0.40) MAPTALDH1A1KDM4ELMNAMEN1
SCHEMBL2003907 0.92 L3MBTL1 (0.41) MAPTPKMGAAALDH1A1S1PR3
SCHEMBL2006836 0.91 MCL1 (0.40) ALDH1A1KDM4ELMNAMEN1KMT2A
SCHEMBL2006280 0.90 FAAH (0.44) MAPTGAAALDH1A1KDM4EMEN1
SCHEMBL2007516 0.89 S1PR3 (0.38) MAPTPKMGAAALDH1A1S1PR3
SCHEMBL2006664 0.88 ALOX5AP (0.36) MAPTPKMGAAALDH1A1S1PR3
SCHEMBL2004791 0.88 MAPT (0.44) MAPTPKMGAAALDH1A1S1PR3
SCHEMBL2006216 0.88 ACHE (0.47) MAPTPKMALDH1A1LMNAMEN1
SCHEMBL2004677 0.88 MAPT (0.41) MAPTPKMGAAALDH1A1S1PR3
SCHEMBL2002167 0.87 ALOX5AP (0.43) MAPTLMNAALOX5APCYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed