SCHEMBL2004791

SCHEMBL2004791

O=C(c1cnc(-c2ccccc2)o1)c1c(Cl)n(Cc2ccc(Cl)cc2)c2ccc(O)cc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.44
ALDH1A1 P00352 3/20 0.44
GAA P10253 2/20 0.44
PKM P14618 2/20 0.44
KDM4E B2RXH2 2/20 0.42
LMNA P02545 2/20 0.42
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
S1PR3 Q99500 2/20 0.41
PTGES2 Q9H7Z7 3/20 0.39
PTGES O14684 1/20 0.39
ALOX5AP P20292 1/20 0.39
PLA2G2A P14555 1/20 0.39
EIF4A3 P38919 2/20 0.39
USP2 O75604 1/20 0.39
POLB P06746 1/20 0.39
TP53 P04637 1/20 0.38
CYP3A4 P08684 2/20 0.38
ALOX15 P16050 1/20 0.38
TSHR P16473 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2012906 0.93 MAPT (0.44) MAPTALDH1A1KDM4ELMNAMEN1
SCHEMBL2007363 0.91 ALOX5AP (0.40) MAPTALDH1A1GAAPKMKDM4E
SCHEMBL2008306 0.91 L3MBTL1 (0.43) MAPTALDH1A1GAAPKMKDM4E
SCHEMBL2003239 0.91 PTGES2 (0.41) MAPTALDH1A1GAAPKMKDM4E
SCHEMBL2002616 0.90 ALDH1A1 (0.45) MAPTALDH1A1KDM4ELMNAMEN1
SCHEMBL2003126 0.90 MEN1 (0.44) ALDH1A1GAAKDM4EMEN1KMT2A
SCHEMBL2005862 0.88 MAPT (0.41) MAPTALDH1A1GAAPKMKDM4E
SCHEMBL1999222 0.88 MAPT (0.40) MAPTALDH1A1GAAPKMKDM4E
SCHEMBL1999556 0.87 PLA2G2A (0.49) MAPTALDH1A1PKMLMNAMEN1
SCHEMBL2004203 0.86 ALOX5AP (0.45) ALDH1A1KDM4EALOX5APPLA2G2ACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed