SCHEMBL1999556

SCHEMBL1999556

COc1ccc2c(c1)c(C(=O)c1cnc(-c3ccccc3)o1)c(Cl)n2Cc1ccc(Cl)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLA2G2A P14555 9/20 0.49
ALDH1A1 P00352 3/20 0.49
TSHR P16473 2/20 0.49
MEN1 O00255 1/20 0.49
RGS12 O14924 1/20 0.49
LMNA P02545 1/20 0.49
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
MAPT P10636 1/20 0.49
CYP2C9 P11712 1/20 0.49
PKM P14618 1/20 0.49
NFKB1 P19838 1/20 0.49
MAPK1 P28482 1/20 0.49
CYP2C19 P33261 1/20 0.49
GNAI1 P63096 1/20 0.49
PMP22 Q01453 1/20 0.49
KMT2A Q03164 1/20 0.49
HIF1A Q16665 1/20 0.49
ACHE P22303 1/20 0.47
PLA2G1B P04054 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2002049 0.92 PLA2G2A (0.58) PLA2G2AALDH1A1TSHRMEN1RGS12
SCHEMBL2004203 0.92 ALOX5AP (0.45) PLA2G2AALDH1A1CYP3A4CYP2C9MAPK1
SCHEMBL2005932 0.92 MEN1 (0.46) PLA2G2AALDH1A1TSHRMEN1RGS12
SCHEMBL2002932 0.92 PLA2G2A (0.43) PLA2G2AALDH1A1TSHRMEN1RGS12
SCHEMBL2002482 0.91 ALDH1A1 (0.44) PLA2G2AALDH1A1TSHRMEN1RGS12
SCHEMBL2012906 0.90 MAPT (0.44) ALDH1A1TSHRMEN1LMNACYP3A4
SCHEMBL2003930 0.89 PLA2G2A (0.46) PLA2G2AALDH1A1TSHRMEN1RGS12
SCHEMBL2006216 0.89 ACHE (0.47) PLA2G2AALDH1A1TSHRMEN1RGS12
SCHEMBL2003126 0.88 MEN1 (0.44) ALDH1A1MEN1KMT2AALOX5AP
SCHEMBL2002896 0.88 PLA2G2A (0.49) PLA2G2AALDH1A1TSHRMEN1RGS12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed