SCHEMBL2002932

SCHEMBL2002932

COc1ccc2c(c1)c(C(=O)c1cnc(-c3ccccc3)o1)c(Cl)n2Cc1ccc(Cl)cc1Cl

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLA2G2A P14555 9/20 0.43
MAPT P10636 3/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
RGS12 O14924 1/20 0.41
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
PKM P14618 1/20 0.41
TSHR P16473 1/20 0.41
NFKB1 P19838 1/20 0.41
MAPK1 P28482 1/20 0.41
CYP2C19 P33261 1/20 0.41
GNAI1 P63096 1/20 0.41
PMP22 Q01453 1/20 0.41
HIF1A Q16665 1/20 0.41
ACHE P22303 1/20 0.41
EDNRB P24530 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2011328 0.93 LMNA (0.40) PLA2G2AMAPTALDH1A1LMNACYP1A2
SCHEMBL2003542 0.93 MAPT (0.39) PLA2G2AMAPTMEN1KMT2ARGS12
SCHEMBL2003889 0.92 ALDH1A1 (0.38) PLA2G2AMAPTMEN1KMT2ARGS12
SCHEMBL1999556 0.92 PLA2G2A (0.49) PLA2G2AMAPTMEN1KMT2ARGS12
SCHEMBL1999686 0.92 MAPT (0.42) MAPTMEN1KMT2AALDH1A1LMNA
SCHEMBL2006531 0.90 PLA2G2A (0.41) PLA2G2AMAPTMEN1KMT2ARGS12
SCHEMBL2008123 0.90 ACHE (0.41) PLA2G2AMAPTMEN1KMT2ARGS12
SCHEMBL2008233 0.89 LMNA (0.39) MAPTMEN1KMT2AALDH1A1LMNA
SCHEMBL2005563 0.89 LMNA (0.45) MAPTMEN1KMT2AALDH1A1LMNA
SCHEMBL2008306 0.88 L3MBTL1 (0.43) MAPTMEN1KMT2AALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed