SCHEMBL2003126

SCHEMBL2003126

Cc1ccc2c(c1)c(C(=O)c1cnc(-c3ccccc3)o1)c(Cl)n2Cc1ccc(Cl)cc1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.44
HTT P42858 1/20 0.44
KMT2A Q03164 1/20 0.44
FAAH O00519 1/20 0.43
PTGES2 Q9H7Z7 6/20 0.43
PTGES O14684 3/20 0.43
ALDH1A1 P00352 2/20 0.42
KDM4E B2RXH2 1/20 0.42
GAA P10253 1/20 0.42
HSD17B10 Q99714 1/20 0.42
CNR2 P34972 2/20 0.41
ALOX5AP P20292 1/20 0.40
PPARG P37231 1/20 0.39
AKR1B1 P15121 1/20 0.39
PTGDR2 Q9Y5Y4 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
ALOX5 P09917 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2012906 0.92 MAPT (0.44) MEN1KMT2APTGES2PTGESALDH1A1
SCHEMBL2001978 0.92 FAAH (0.45) MEN1HTTKMT2AFAAHPTGES2
SCHEMBL2008233 0.91 LMNA (0.39) MEN1HTTKMT2AFAAHPTGES2
SCHEMBL2002956 0.91 PTGES2 (0.44) MEN1HTTKMT2AFAAHPTGES2
SCHEMBL2004791 0.90 MAPT (0.44) MEN1KMT2APTGES2PTGESALDH1A1
SCHEMBL2002616 0.89 ALDH1A1 (0.45) MEN1KMT2APTGES2ALDH1A1KDM4E
SCHEMBL2010143 0.88 PTGES2 (0.42) MEN1HTTKMT2AFAAHPTGES2
SCHEMBL2006280 0.88 FAAH (0.44) MEN1HTTKMT2AFAAHPTGES2
SCHEMBL1999556 0.88 PLA2G2A (0.49) MEN1KMT2AALDH1A1ALOX5AP
SCHEMBL2004203 0.87 ALOX5AP (0.45) ALDH1A1KDM4EHSD17B10ALOX5APALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed